U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 16:11:40 UTC 2023
Edited
by admin
on Sat Dec 16 16:11:40 UTC 2023
Protein Type MONOCLONAL ANTIBODY
Protein Sub Type IGG1
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
M9SE4M9U1V
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
BARECETAMAB
INN  
Official Name English
IMMUNOGLOBULIN G1-LAMBDA, ANTI-(HOMO SAPIENS ERBB3 (RECEPTOR TYROSINE-PROTEIN KINASE ERBB-3, HER3)), HOMO SAPIENS MONOCLONAL ANTIBODY; GAMMA1 HEAVY CHAIN HOMO SAPIENS (1-451) (VH (HOMO SAPIENS IGHV3-23*01 (90.8%)-(IGHD)-IGHJ4*01 (100%)) CDR-IMGT (8.8.14)
Common Name English
Barecetamab [WHO-DD]
Common Name English
ISU104
Code English
barecetamab [INN]
Common Name English
ISU-104
Code English
IMMUNOGLOBULIN G1, ANTI-(HUMAN EPIDERMAL GROWTH FACTOR RECEPTOR HER3) (HUMAN MONOCLONAL ISU104 .GAMMA.1-CHAIN), DISULFIDE WITH HUMAN MONOCLONAL ISU104 .LAMBDA.-CHAIN, DIMER
Common Name English
Code System Code Type Description
NCI_THESAURUS
C158746
Created by admin on Sat Dec 16 16:11:40 UTC 2023 , Edited by admin on Sat Dec 16 16:11:40 UTC 2023
PRIMARY
INN
11386
Created by admin on Sat Dec 16 16:11:40 UTC 2023 , Edited by admin on Sat Dec 16 16:11:40 UTC 2023
PRIMARY
FDA UNII
M9SE4M9U1V
Created by admin on Sat Dec 16 16:11:40 UTC 2023 , Edited by admin on Sat Dec 16 16:11:40 UTC 2023
PRIMARY
CAS
2275727-74-5
Created by admin on Sat Dec 16 16:11:40 UTC 2023 , Edited by admin on Sat Dec 16 16:11:40 UTC 2023
PRIMARY
From To
4_138 4_197
4_22 4_89
3_138 3_197
3_22 3_89
2_371 2_429
2_265 2_325
2_224 4_215
2_148 2_204
2_22 2_96
1_371 1_429
1_265 1_325
1_233 2_233
1_230 2_230
1_224 3_215
1_148 1_204
1_22 1_96
Glycosylation Link Type Site
N 1_301
N 2_301
Related Record Type Details
TARGET -> INHIBITOR
ISU104 completely suppressed Heregulin HRG-induced phosphorylation
Related Record Type Details
ACTIVE MOIETY
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL