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Details

Stereochemistry ABSOLUTE
Molecular Formula C51H60N3O11S.3Na
Molecular Weight 992.07
Optical Activity UNSPECIFIED
Defined Stereocenters 12 / 12
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of FLUORESCEIN LISICOL TRISODIUM

SMILES

[Na+].[Na+].[Na+].C[C@H](CCC(=O)N[C@@H](CCCCNC(=S)NC1=CC=C2C(=C1)C(=O)OC23C4=CC=C([O-])C=C4OC5=C3C=CC([O-])=C5)C([O-])=O)[C@H]6CC[C@H]7[C@@H]8[C@H](O)C[C@@H]9C[C@H](O)CC[C@]9(C)[C@H]8C[C@H](O)[C@]67C

InChI

InChIKey=QVHBTANNAWPFGJ-MILHWSGHSA-K
InChI=1S/C51H63N3O11S.3Na/c1-26(33-14-15-37-45-38(25-43(59)50(33,37)3)49(2)18-17-31(57)20-27(49)21-40(45)58)7-16-44(60)54-39(46(61)62)6-4-5-19-52-48(66)53-28-8-11-34-32(22-28)47(63)65-51(34)35-12-9-29(55)23-41(35)64-42-24-30(56)10-13-36(42)51;;;/h8-13,22-24,26-27,31,33,37-40,43,45,55-59H,4-7,14-21,25H2,1-3H3,(H,54,60)(H,61,62)(H2,52,53,66);;;/q;3*+1/p-3/t26-,27+,31-,33-,37+,38+,39+,40-,43+,45+,49+,50-;;;/m1.../s1

HIDE SMILES / InChI

Molecular Formula C51H60N3O11S
Molecular Weight 923.101
Charge -3
Count
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 12 / 12
E/Z Centers 0
Optical Activity UNSPECIFIED

Molecular Formula Na
Molecular Weight 22.98976928
Charge 1
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Fluorescein Lisicol (NRL972) is a fluorescent-labelled bile acid analog that is used as an investigational marker for liver function, specifically hepatic biliary transporter function. Fluorescein Lisicol has been used in trials investigating the pharmacokinetics of hepatic cirrhosis, viral hepatitis, non-alcoholic steatohepatitis and non-alcoholic fatty liver disease.

Approval Year

PubMed

PubMed

TitleDatePubMed
Effects of renal insufficiency on the elimination of fluorescein lisicol (NRL972), an investigational marker of hepatic transporter function.
2015-07
Gateways to clinical trials.
2004-09
Substance Class Chemical
Created
by admin
on Tue Apr 01 22:27:55 GMT 2025
Edited
by admin
on Tue Apr 01 22:27:55 GMT 2025
Record UNII
LV71380AGP
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
L-LYSINE, N6-(((3',6'-DIHYDROXY-3-OXOSPIRO(ISOBENZOFURAN-1(3H),9'-(9H)XANTHEN)-5-YL)AMINO)THIOXOMETHYL)-N2-((3.ALPHA.,5.BETA.,7.ALPHA.,12.ALPHA.)-3,7,12-TRIHYDROXY-24-OXOCHOLAN-24-YL)-, TRISODIUM SALT
Preferred Name English
FLUORESCEIN LISICOL TRISODIUM
Common Name English
FLUORESCEIN LISICOL TRISODIUM SALT
Common Name English
NRL-972 TRISODIUM
Code English
Code System Code Type Description
CAS
463932-51-6
Created by admin on Tue Apr 01 22:27:55 GMT 2025 , Edited by admin on Tue Apr 01 22:27:55 GMT 2025
ALTERNATIVE
PUBCHEM
134819855
Created by admin on Tue Apr 01 22:27:55 GMT 2025 , Edited by admin on Tue Apr 01 22:27:55 GMT 2025
PRIMARY
FDA UNII
LV71380AGP
Created by admin on Tue Apr 01 22:27:55 GMT 2025 , Edited by admin on Tue Apr 01 22:27:55 GMT 2025
PRIMARY
CAS
397841-88-2
Created by admin on Tue Apr 01 22:27:55 GMT 2025 , Edited by admin on Tue Apr 01 22:27:55 GMT 2025
PRIMARY
Related Record Type Details
PARENT -> SALT/SOLVATE
Related Record Type Details
ACTIVE MOIETY