U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 12:19:08 UTC 2023
Edited
by admin
on Sat Dec 16 12:19:08 UTC 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
LR4LA8YD5Z
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
BROMODOMAIN-CONTAINING PROTEIN 2
Common Name English
RING3
Common Name English
REALLY INTERESTING NEW GENE 3 PROTEIN
Common Name English
KIAA9001
Common Name English
O27.1.1
Common Name English
BRD2
Common Name English
Code System Code Type Description
UNIPROT
P25440
Created by admin on Sat Dec 16 12:19:08 UTC 2023 , Edited by admin on Sat Dec 16 12:19:08 UTC 2023
PRIMARY
FDA UNII
LR4LA8YD5Z
Created by admin on Sat Dec 16 12:19:08 UTC 2023 , Edited by admin on Sat Dec 16 12:19:08 UTC 2023
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
BRD2(BD2) DOMAIN
Kd
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Kd
INHIBITOR -> TARGET
A >250x differential binding preference for BDII over BDI
BINDING
INHIBITOR -> TARGET
IC50
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL