U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:53:48 GMT 2025
Edited
by admin
on Tue Apr 01 16:53:48 GMT 2025
Protein Type ENZYME
Protein Sub Type SERINE/THREONINE-PROTEIN KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
LC31QDE6K8
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
DARDARIN
Preferred Name English
LEUCINE-RICH REPEAT SERINE/THREONINE-PROTEIN KINASE 2
Common Name English
LRRK2
Common Name English
PARK8
Common Name English
Code System Code Type Description
FDA UNII
LC31QDE6K8
Created by admin on Tue Apr 01 16:53:48 GMT 2025 , Edited by admin on Tue Apr 01 16:53:48 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
DNL151 is a selective, orally bioavailable, central nervous system–penetrant, reversible inhibitor of leucine-rich repeat kinase 2 (LRRK2)
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_935] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL