U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
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Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:44:57 GMT 2025
Edited
by admin
on Tue Apr 01 16:44:57 GMT 2025
Protein Type RECEPTOR
Protein Sub Type G PROTEIN-COUPLED RECEPTOR
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
L5QY0GLC6X
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
Endothelin receptor type B
Common Name English
ENDOTHELIN B RECEPTOR
Preferred Name English
ET-B
Common Name English
ET-BR
Common Name English
ETRB
Common Name English
ENDOTHELIN RECEPTOR NON-SELECTIVE TYPE
Common Name English
Code System Code Type Description
FDA UNII
L5QY0GLC6X
Created by admin on Tue Apr 01 16:44:57 GMT 2025 , Edited by admin on Tue Apr 01 16:44:57 GMT 2025
PRIMARY
UNIPROT
P24530
Created by admin on Tue Apr 01 16:44:57 GMT 2025 , Edited by admin on Tue Apr 01 16:44:57 GMT 2025
PRIMARY
PHAROS
P24530
Created by admin on Tue Apr 01 16:44:57 GMT 2025 , Edited by admin on Tue Apr 01 16:44:57 GMT 2025
PRIMARY
From To
1_148 1_229
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_33
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
WEAK INHIBITOR->OFF TARGET
Porcine cerebellum membranes.
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_376] [1_377] [1_379] S-PALMITOYL CYSTEINE 08WQ73S7SV
AMINO_ACID_SUBSTITUTION [1_279] [1_393] [1_414] [1_415] [1_416] DEXFOSFOSERINE VI4F0K069V
AMINO_ACID_SUBSTITUTION [1_413] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL