Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:52:13 GMT 2025
by
admin
on
Tue Apr 01 16:52:13 GMT 2025
|
Protein Sub Type | |
Sequence Type | COMPLETE |
Record UNII |
L01TYM08QX
|
Record Status |
Validated (UNII)
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Record Version |
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-
Download
Name | Type | Language | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
Code System | Code | Type | Description | ||
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P22607
Created by
admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
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PRIMARY | |||
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P22607
Created by
admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
|
PRIMARY | |||
|
L01TYM08QX
Created by
admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
|
PRIMARY |
From | To |
---|---|
1_39 | 1_87 |
1_154 | 1_206 |
1_253 | 1_317 |
Glycosylation Type | HUMAN |
Glycosylation Link Type | Site |
---|---|
N | 1_76 |
N | 1_203 |
N | 1_240 |
N | 1_272 |
N | 1_293 |
N | 1_306 |
Related Record | Type | Details | ||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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MUTANT->PARENT |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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DERIVATIVE -> PARENT | |||
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CONJUGATED TOXIN->TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
at higher concentrations that were still clinically achievable
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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Structural Modifications
Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
---|---|---|---|---|---|---|
AMINO ACID SUBSTITUTION | [1_422] [1_423] | DEXFOSFOSERINE | VI4F0K069V | |||
AMINO ACID SUBSTITUTION | [1_625] [1_626] [1_702] [1_738] | TYROSINE O-PHOSPHATE | 2R86C98KDX |
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
MOL_WEIGHT | CHEMICAL |
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Molecular Formula | CHEMICAL |
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