U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
This repository is under review for potential modification in compliance with Administration directives.

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:52:13 GMT 2025
Edited
by admin
on Tue Apr 01 16:52:13 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
L01TYM08QX
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
FGFR-3
Preferred Name English
FIBROBLAST GROWTH FACTOR RECEPTOR 3
Common Name English
JTK4
Common Name English
FGFR3
Common Name English
Code System Code Type Description
PHAROS
P22607
Created by admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
PRIMARY
UNIPROT
P22607
Created by admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
PRIMARY
FDA UNII
L01TYM08QX
Created by admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
PRIMARY
From To
1_39 1_87
1_154 1_206
1_253 1_317
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_76
N 1_203
N 1_240
N 1_272
N 1_293
N 1_306
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
MUTANT->PARENT
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
DERIVATIVE -> PARENT
CONJUGATED TOXIN->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
at higher concentrations that were still clinically achievable
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_422] [1_423] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_625] [1_626] [1_702] [1_738] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL