Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 21:03:10 GMT 2025
by
admin
on
Tue Apr 01 21:03:10 GMT 2025
|
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
KDM3YPI7TR
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| Record Status |
Validated (UNII)
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| Record Version |
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-
Download
| Name | Type | Language | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
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KDM3YPI7TR
Created by
admin on Tue Apr 01 21:03:10 GMT 2025 , Edited by admin on Tue Apr 01 21:03:10 GMT 2025
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PRIMARY | |||
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Q92793
Created by
admin on Tue Apr 01 21:03:10 GMT 2025 , Edited by admin on Tue Apr 01 21:03:10 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
Inhibits binding of CREB to Catenin beta-1 and CREB binding protein (CBP)/ -catenin signaling
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
![Structure of (6S,9aS)-N-benzyl-6-(4-hydroxybenzyl)-4,7-dioxo-2-((3-(pyridin-2-yl)isoxazol-5-yl)methyl)-8-(quinolin-5-ylmethyl)hexahydro-2H-pyrazino[2,1-c][1,2,4]triazine-1(6H)-carboxamide](/img/189bdc67-6df3-402d-8520-2c80005047f8.svg "Structure of (6S,9aS)-N-benzyl-6-(4-hydroxybenzyl)-4,7-dioxo-2-((3-(pyridin-2-yl)isoxazol-5-yl)methyl)-8-(quinolin-5-ylmethyl)hexahydro-2H-pyrazino[2,1-c][1,2,4]triazine-1(6H)-carboxamide")
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO_ACID_SUBSTITUTION | [1_120] [1_1029] [1_1381] [1_1385] [1_1762] [1_2062] [1_2075] [1_2078] [1_2350] | DEXFOSFOSERINE | VI4F0K069V | |||
| AMINO_ACID_SUBSTITUTION | [1_1] | N-ACETYLALANINE | 26C4VY6Z0M | |||
| AMINO_ACID_SUBSTITUTION | [1_219] [1_600] [1_624] | TILARGININE | 27JT06E6GR | |||
| AMINO_ACID_SUBSTITUTION | [1_656] [1_1013] [1_1215] [1_1582] [1_1590] [1_1591] [1_1596] [1_1740] [1_1743] | N6-ACETYLLYSINE | 470AD5VY1X |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
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