U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 16:17:04 GMT 2025
Edited
by admin
on Wed Apr 02 16:17:04 GMT 2025
Protein Type RECEPTOR
Protein Sub Type KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
K33ESJ3L25
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
HIGH AFFINITY NERVE GROWTH FACTOR RECEPTOR G595R
Common Name English
TRKA G595R
Preferred Name English
TYROSINE KINASE RECEPTOR A G595R
Common Name English
TROPOMYOSIN RECEPTOR KINASE A G595R MUTANT
Common Name English
Code System Code Type Description
FDA UNII
K33ESJ3L25
Created by admin on Wed Apr 02 16:17:04 GMT 2025 , Edited by admin on Wed Apr 02 16:17:04 GMT 2025
PRIMARY
From To
1_122 1_159
1_183 1_233
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_35
N 1_63
N 1_89
N 1_156
N 1_170
N 1_221
N 1_230
N 1_249
N 1_286
N 1_291
N 1_306
N 1_326
N 1_369
Related Record Type Details
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_464] [1_644] [1_648] [1_649] [1_759] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL