Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Sat Dec 16 12:05:23 GMT 2023
by
admin
on
Sat Dec 16 12:05:23 GMT 2023
|
Protein Sub Type | |
Sequence Origin | HUMAN |
Sequence Type | COMPLETE |
Record UNII |
JS20X60RRY
|
Record Status |
Validated (UNII)
|
Record Version |
|
-
Download
Name | Type | Language | ||
---|---|---|---|---|
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
Code System | Code | Type | Description | ||
---|---|---|---|---|---|
|
SYK
Created by
admin on Sat Dec 16 12:05:24 GMT 2023 , Edited by admin on Sat Dec 16 12:05:24 GMT 2023
|
PRIMARY | |||
|
P43405
Created by
admin on Sat Dec 16 12:05:24 GMT 2023 , Edited by admin on Sat Dec 16 12:05:24 GMT 2023
|
PRIMARY | |||
|
JS20X60RRY
Created by
admin on Sat Dec 16 12:05:24 GMT 2023 , Edited by admin on Sat Dec 16 12:05:24 GMT 2023
|
PRIMARY | |||
|
P43405
Created by
admin on Sat Dec 16 12:05:24 GMT 2023 , Edited by admin on Sat Dec 16 12:05:24 GMT 2023
|
PRIMARY |
Related Record | Type | Details | ||
---|---|---|---|---|
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
Assessed by Invitrogen/Life Technologies using the Z’-LYTE assay format
REVERSIBLE
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
Dropped from clinical trials because of adverse events probably bleeding.
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
inhibited its kinase activity as an ATP-competitive inhibitor (Ki = 30 nM)
COMPETITIVE INHIBITOR
Ki
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
Molecular Formula | CHEMICAL |
|
||||
MOL_WEIGHT | CHEMICAL |
|