U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 19:21:45 GMT 2025
Edited
by admin
on Tue Apr 01 19:21:45 GMT 2025
Protein Type ENZYME
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
J8U2X4699C
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
AP2-ASSOCIATED PROTEIN KINASE 1
Common Name English
AAK1
Preferred Name English
KIAA1048
Common Name English
ADAPTOR-ASSOCIATED KINASE 1
Common Name English
Code System Code Type Description
CAS
444185-98-2
Created by admin on Tue Apr 01 19:21:45 GMT 2025 , Edited by admin on Tue Apr 01 19:21:45 GMT 2025
GENERIC (FAMILY)
PHAROS
Q2M2I8
Created by admin on Tue Apr 01 19:21:45 GMT 2025 , Edited by admin on Tue Apr 01 19:21:45 GMT 2025
PRIMARY
FDA UNII
J8U2X4699C
Created by admin on Tue Apr 01 19:21:45 GMT 2025 , Edited by admin on Tue Apr 01 19:21:45 GMT 2025
PRIMARY
UNIPROT
Q2M2I8
Created by admin on Tue Apr 01 19:21:45 GMT 2025 , Edited by admin on Tue Apr 01 19:21:45 GMT 2025
PRIMARY
WIKIPEDIA
AAK1
Created by admin on Tue Apr 01 19:21:45 GMT 2025 , Edited by admin on Tue Apr 01 19:21:45 GMT 2025
PRIMARY
EC (ENZYME CLASS)
EC 2.7.11.1
Created by admin on Tue Apr 01 19:21:45 GMT 2025 , Edited by admin on Tue Apr 01 19:21:45 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
CELL ASSAY
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_14] [1_235] [1_618] [1_623] [1_624] [1_637] [1_650] [1_731] [1_846] [1_937] [1_938] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL