U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 14:56:30 UTC 2023
Edited
by admin
on Sat Dec 16 14:56:30 UTC 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
J35DH4R1TA
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
HIGH AFFINITY CAMP-SPECIFIC 3',5'-CYCLIC PHOSPHODIESTERASE 7A
Common Name English
TM22
Common Name English
PDE7A
Common Name English
HCP1
Common Name English
Code System Code Type Description
PHAROS
Q13946
Created by admin on Sat Dec 16 14:56:30 UTC 2023 , Edited by admin on Sat Dec 16 14:56:30 UTC 2023
PRIMARY
UNIPROT
Q13946
Created by admin on Sat Dec 16 14:56:30 UTC 2023 , Edited by admin on Sat Dec 16 14:56:30 UTC 2023
PRIMARY
FDA UNII
J35DH4R1TA
Created by admin on Sat Dec 16 14:56:30 UTC 2023 , Edited by admin on Sat Dec 16 14:56:30 UTC 2023
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
Selective PDE7 inhibitor. Percent inhibition of other PDEs (PDE1A, 3A, 5A, 6, 8A1, 9A2, and 11A4) by 1 μM of MTP38 were less than 50%.
IC50
INHIBITOR -> TARGET
INHIBITOR OF EXPRESSION->TARGET
RADIOLIGAND->TARGET
Selective PDE7 inhibitor. Percent inhibition of other PDEs (PDE1A, 3A, 5A, 6, 8A1, 9A2, and 11A4) by 1 μM of MTP38 were less than 50%.
IC50
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL