Details
| Stereochemistry | ABSOLUTE |
| Molecular Formula | C16H24N2O3.ClH |
| Molecular Weight | 328.834 |
| Optical Activity | UNSPECIFIED |
| Defined Stereocenters | 1 / 1 |
| E/Z Centers | 0 |
| Charge | 0 |
SHOW SMILES / InChI
SMILES
Cl.CC(C)(C)NC[C@@H](O)COC1=C2CCC(=O)NC2=CC=C1
InChI
InChIKey=FYBXRCFPOTXTJF-RFVHGSKJSA-N
InChI=1S/C16H24N2O3.ClH/c1-16(2,3)17-9-11(19)10-21-14-6-4-5-13-12(14)7-8-15(20)18-13;/h4-6,11,17,19H,7-10H2,1-3H3,(H,18,20);1H/t11-;/m1./s1
| Molecular Formula | C16H24N2O3 |
| Molecular Weight | 292.3734 |
| Charge | 0 |
| Count |
|
| Stereochemistry | ABSOLUTE |
| Additional Stereochemistry | No |
| Defined Stereocenters | 1 / 1 |
| E/Z Centers | 0 |
| Optical Activity | UNSPECIFIED |
| Molecular Formula | ClH |
| Molecular Weight | 36.461 |
| Charge | 0 |
| Count |
|
| Stereochemistry | ACHIRAL |
| Additional Stereochemistry | No |
| Defined Stereocenters | 0 / 0 |
| E/Z Centers | 0 |
| Optical Activity | NONE |
(R)-Carteolol is an enantiomer of the drug carteolol that is used to treat glaucoma. (R)-Carteolol is a partial agonist with the high affinity to the beta-adrenoceptors. It was shown, that in the treatment of glaucoma, the therapeutic advantage of the R(+)-isomers is similar to the S(-)-isomers and there is no stereoselectivity between the two enantiomers.
Approval Year
PubMed
| Title | Date | PubMed |
|---|---|---|
| Effects of the R(+)- and S(-)-isomers of beta-adrenoceptor blockers with intrinsic sympathomimetic activity, befunolol and carteolol, on rabbit intraocular pressure. | 1991-08 |
|
| Comparison of interactions of R-(+)- and S-(-)-isomers of beta-adrenergic partial agonists, befunolol and carteolol, with high affinity site of beta-adrenoceptors in isolated rabbit ciliary body and guinea-pig taenia caeci. | 1991-07 |
| Substance Class |
Chemical
Created
by
admin
on
Edited
Mon Mar 31 23:31:39 GMT 2025
by
admin
on
Mon Mar 31 23:31:39 GMT 2025
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| Record UNII |
IN6W2DDZ31
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| Record Status |
Validated (UNII)
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| Record Version |
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Common Name | English |
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59567-87-2
Created by
admin on Mon Mar 31 23:31:39 GMT 2025 , Edited by admin on Mon Mar 31 23:31:39 GMT 2025
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IN6W2DDZ31
Created by
admin on Mon Mar 31 23:31:39 GMT 2025 , Edited by admin on Mon Mar 31 23:31:39 GMT 2025
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12285396
Created by
admin on Mon Mar 31 23:31:39 GMT 2025 , Edited by admin on Mon Mar 31 23:31:39 GMT 2025
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| Related Record | Type | Details | ||
|---|---|---|---|---|
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RACEMATE -> ENANTIOMER |
