Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 23:50:56 GMT 2025
by
admin
on
Tue Apr 01 23:50:56 GMT 2025
|
Protein Type | ENZYME |
Protein Sub Type | SERINE/THREONINE-PROTEIN KINASE |
Sequence Origin | HUMAN |
Sequence Type | COMPLETE |
Record UNII |
IEQ8K30M47
|
Record Status |
Validated (UNII)
|
Record Version |
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-
Download
Name | Type | Language | ||
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Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
Code System | Code | Type | Description | ||
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IEQ8K30M47
Created by
admin on Tue Apr 01 23:50:56 GMT 2025 , Edited by admin on Tue Apr 01 23:50:56 GMT 2025
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PRIMARY | |||
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P24941
Created by
admin on Tue Apr 01 23:50:56 GMT 2025 , Edited by admin on Tue Apr 01 23:50:56 GMT 2025
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PRIMARY |
Related Record | Type | Details | ||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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WEAK INHIBITOR->TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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||
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INHIBITOR -> TARGET |
IC50
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||
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INHIBITOR -> TARGET |
IC50
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||
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INHIBITOR -> TARGET |
IC50
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||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
Selective inhibitor
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
The development of bronchopulmonary hemorrhage and sepsis resulted in the death of two patients. The study was ultimately terminated prematurely due to an unfavorable risk-benefit ratio in patients.
IC50
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WEAK INHIBITOR->TARGET |
IC50
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Structural Modifications
Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
---|---|---|---|---|---|---|
AMINO_ACID_SUBSTITUTION | [1_14] [1_160] | SITE_SPECIFIC | THREONINE PHOSPHATE | 3L4WX7B1EI | ||
AMINO_ACID_SUBSTITUTION | [1_15] [1_19] | SITE_SPECIFIC | TYROSINE O-PHOSPHATE | 2R86C98KDX | ||
AMINO_ACID_SUBSTITUTION | [1_6] | SITE_SPECIFIC | N6-ACETYLLYSINE | 470AD5VY1X | ||
AMINO_ACID_SUBSTITUTION | [1_1] | SITE_SPECIFIC | N-ACETYLMETHIONINE | 9J12WX5B6A |
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
MOL_WEIGHT | CHEMICAL |
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