U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 16:43:19 GMT 2025
Edited
by admin
on Wed Apr 02 16:43:19 GMT 2025
Protein Type STRUCTURAL PROTEIN
Protein Sub Type TUBULIN
Record UNII
GK82JF3ZU4
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
TUBULIN ALPHA-BETA DIMER
Common Name English
TUBULIN DIMER
Preferred Name English
Code System Code Type Description
FDA UNII
GK82JF3ZU4
Created by admin on Wed Apr 02 16:43:19 GMT 2025 , Edited by admin on Wed Apr 02 16:43:19 GMT 2025
PRIMARY
UNIPROT
P07437
Created by admin on Wed Apr 02 16:43:19 GMT 2025 , Edited by admin on Wed Apr 02 16:43:19 GMT 2025
PRIMARY
UNIPROT
Q71U36
Created by admin on Wed Apr 02 16:43:19 GMT 2025 , Edited by admin on Wed Apr 02 16:43:19 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR OF AGGREGATION->TARGET
Sabizabulin binds to the colchicine-binding site of alpha- and beta-tubulin subunits of microtubules and crosslinks the microtubules, thereby inhibiting microtubule polymerization in tumor blood vessel endothelial cells and tumor cells.
IRREVERSIBLE INHIBITOR
INHIBITOR OF AGGREGATION->TARGET
INHIBITOR OF AGGREGATION->TARGET
INHIBITOR OF AGGREGATION->TARGET
BLOCKS OR DESTABILIZED TUBULIN POLYMERS
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL