Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Mon Mar 31 22:33:28 GMT 2025
by
admin
on
Mon Mar 31 22:33:28 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
G53298VN9Y
|
| Record Status |
Validated (UNII)
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| Record Version |
|
-
Download
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| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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DB05599
Created by
admin on Mon Mar 31 22:33:28 GMT 2025 , Edited by admin on Mon Mar 31 22:33:28 GMT 2025
|
PRIMARY | |||
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62031-54-3
Created by
admin on Mon Mar 31 22:33:28 GMT 2025 , Edited by admin on Mon Mar 31 22:33:28 GMT 2025
|
GENERIC (FAMILY) | |||
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G53298VN9Y
Created by
admin on Mon Mar 31 22:33:28 GMT 2025 , Edited by admin on Mon Mar 31 22:33:28 GMT 2025
|
PRIMARY | |||
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m5371
Created by
admin on Mon Mar 31 22:33:28 GMT 2025 , Edited by admin on Mon Mar 31 22:33:28 GMT 2025
|
PRIMARY | Merck Index | ||
|
1591916
Created by
admin on Mon Mar 31 22:33:28 GMT 2025 , Edited by admin on Mon Mar 31 22:33:28 GMT 2025
|
PRIMARY | RxNorm | ||
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G53298VN9Y
Created by
admin on Mon Mar 31 22:33:28 GMT 2025 , Edited by admin on Mon Mar 31 22:33:28 GMT 2025
|
PRIMARY | |||
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106096-92-8
Created by
admin on Mon Mar 31 22:33:28 GMT 2025 , Edited by admin on Mon Mar 31 22:33:28 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR -> TARGET |
Prevents FGFR ligands, such as FGF1, FGF2, FGF4, from binding to their cognate receptors, thereby inhibiting the activation of the related FGFR tyrosine kinases. Inhibition of FGFR1 by this agent may retard tumor cell proliferation and induce tumor cell death. FP-1039 may also inhibit vascular endothelial growth factor (VEGF)-induced angiogenesis. FGFR1 is a receptor tyrosine kinase upregulated in certain tumor cells and involved in tumor cellular proliferation, differentiation, angiogenesis, and survival; most ligands that bind to FGFR1 also bind to the related receptors FGFR3 and FGFR4.
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LIGAND->TARGET |
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| Related Record | Type | Details | ||
|---|---|---|---|---|
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ACTIVE MOIETY |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
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| Molecular Formula | CHEMICAL |
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