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Details

Stereochemistry ACHIRAL
Molecular Formula C7H6N2
Molecular Weight 118.1359
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of IMIDAZO(1,2-A)PYRIDINE

SMILES

C1=CN2C=CC=CC2=N1

InChI

InChIKey=UTCSSFWDNNEEBH-UHFFFAOYSA-N
InChI=1S/C7H6N2/c1-2-5-9-6-4-8-7(9)3-1/h1-6H

HIDE SMILES / InChI

Molecular Formula C7H6N2
Molecular Weight 118.1359
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Approval Year

PubMed

PubMed

TitleDatePubMed
Post Groebke-Blackburn multicomponent protocol: synthesis of new polyfunctional imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrimidine derivatives as potential antimicrobial agents.
2010-12
Ethyl 8-(4-nitro-phen-yl)imidazo[1,2-a]pyridine-7-carboxyl-ate.
2010-11-24
Pharmacophore modeling and 3D-QSAR analysis of phosphoinositide 3-kinase p110alpha inhibitors.
2010-09
Intra-periaqueductal grey microinjections of an imidazo[1,2-b]pyridazine derivative, DM2, affects rostral ventromedial medulla cell activity and shows antinociceptive effect.
2010-03
Modulation of carcinogen metabolizing enzymes by new fused heterocycles pendant to 5,6,7,8-tetrahydronaphthalene derivatives.
2010-02
Efficient one-pot synthetic protocols for iminosugar-bearing imidazo[1,2-a]pyridines from carbohydrates.
2010-01-26
3-(3-Aryloxyaryl)imidazo[1,2-a]pyridine sulfones as liver X receptor agonists.
2010-01-15
Palladium complexes of abnormal N-heterocyclic carbenes as precatalysts for the much preferred Cu-free and amine-free Sonogashira coupling in air in a mixed-aqueous medium.
2009-12-21
Novel one-pot three component reaction for the synthesis of [2-(alkylsulfanyl)imidazo[1,2-a]pyridin-3-yl](aryl)methanone.
2009-11-13
Structure-activity relationship study of EphB3 receptor tyrosine kinase inhibitors.
2009-11-01
Physicochemical properties and membrane interactions of anti-apoptotic derivatives 2-(4-fluorophenyl)-3-(pyridin-4-yl)imidazo[1,2-a]pyridine depending on the hydroxyalkylamino side chain length and conformation: an NMR and ESR study.
2009-09
[5-(2-Fur-yl)-6-nitro-1,2,3,5,6,7-hexa-hydro-imidazo[1,2-a]pyridin-8-yl](phen-yl)methanone.
2009-08-29
Discovery of imidazo[1,2-a]pyridines as potent MCH1R antagonists.
2009-08-15
Orally active C-6 heteroaryl- and heterocyclyl-substituted imidazo[1,2-a]pyridine acid pump antagonists (APAs).
2009-07-01
1-(2-Methyl-imidazo[1,2-a]pyridin-3-yl)-3,3-bis-(methyl-sulfan-yl)prop-2-enone monohydrate.
2009-06-27
Phosphonocarboxylates inhibit the second geranylgeranyl addition by Rab geranylgeranyl transferase.
2009-03-13
Discovery and optimization of imidazo[1,2-a]pyridine inhibitors of insulin-like growth factor-1 receptor (IGF-1R).
2009-02-01
DNA gyrase (GyrB)/topoisomerase IV (ParE) inhibitors: synthesis and antibacterial activity.
2009-02-01
IRAK-4 inhibitors for inflammation.
2009
Synthesis and anticandidal activity of some imidazopyridine derivatives.
2008-12
Chemical-genetic profiling of imidazo[1,2-a]pyridines and -pyrimidines reveals target pathways conserved between yeast and human cells.
2008-11
Synthesis and antituberculosis activity of new hydrazide derivatives.
2008-11
Novel imidazo[1,2-a]naphthyridinic systems (part 1): synthesis, antiproliferative and DNA-intercalating activities.
2008-11
IRAK-4 inhibitors. Part III: a series of imidazo[1,2-a]pyridines.
2008-06-15
IRAK-4 inhibitors. Part II: a structure-based assessment of imidazo[1,2-a]pyridine binding.
2008-06-01
2-Phenyl-imidazo[1,2-a]pyridine-3-carbaldehyde.
2008-04-26
N-(2-Phenyl-imidazo[1,2-a]pyridin-3-yl)acetamide.
2008-04-26
Imidazo[1,2-a]pyridine derivatives as inhibitors of TNF-alpha expression in T cells.
2008-02-01
Switching of polymorph-dependent ESIPT luminescence of an imidazo[1,2-a]pyridine derivative.
2008
Diversification of the three-component coupling of 2-aminoheterocycles, aldehydes, and isonitriles: efficient parallel synthesis of a diverse and druglike library of imidazo- and tetrahydroimidazo[1,2-a] heterocycles.
2007-09-11
Synthesis and biological evaluation of sulfonylhydrazone-substituted imidazo[1,2-a]pyridines as novel PI3 kinase p110alpha inhibitors.
2007-09-01
Recent progress in the pharmacology of imidazo[1,2-a]pyridines.
2007-09
Synthesis and SAR studies of potent imidazopyridine anticoccidial agents.
2007-07-01
Efficient solid-phase synthesis of a library of imidazo[1,2-a]pyridine-8-carboxamides.
2007-02-27
Synthesis and biological evaluation of imidazo[1,2-a]pyridine derivatives as novel PI3 kinase p110alpha inhibitors.
2007-01-01
A novel series of imidazo[1,2-a]pyridine derivatives as HIF-1alpha prolyl hydroxylase inhibitors.
2006-11-01
Synthesis and evaluation of two 18F-labeled imidazo[1,2-a]pyridine analogues as potential agents for imaging beta-amyloid in Alzheimer's disease.
2006-06-01
The cellular phenotype of AZ703, a novel selective imidazo[1,2-a]pyridine cyclin-dependent kinase inhibitor.
2006-03
AZ703, an imidazo[1,2-a]pyridine inhibitor of cyclin-dependent kinases 1 and 2, induces E2F-1-dependent apoptosis enhanced by depletion of cyclin-dependent kinase 9.
2006-01-01
Synthesis of indeno-fused derivatives of quinolizinium salts, imidazo[1,2-a]pyridine, pyrido[1,2-a]indole, and 4h-quinolizin-4-one via benzannulated enyne-allenes.
2005-08-19
Fused heterocycles: synthesis of some new imidazo[1,2-a]- pyridine derivatives.
2004-09-30
Identification of photoproducts from imazosulfuron by HPLC.
2004-09
Studies on the synthesis and characterization of four trans-planaramineplatinum(II) complexes of the form trans-PtL(NH3)CL2 where L = 2-hydroxypyridine, 3-hydroxypyridine, imidazole, and imidazo(1,2-alpha)pyridine.
2004-08
Phenylpiperazinylmethylheterocycle derivatives: synthesis and dopamine receptor binding profiles.
2004-07
Imidazo[1,2-b]pyridazines: a potent and selective class of cyclin-dependent kinase inhibitors.
2004-05-03
Imidazo[1,2-a]pyridines. Part 2: SAR and optimisation of a potent and selective class of cyclin-dependent kinase inhibitors.
2004-05-03
Design and synthesis of acyclic nucleoside analogs with chlorinated imidazo[1,2-a]pyridine bases.
2003-10
Imidazo[1,2-a]pyridines: a potent and selective class of cyclin-dependent kinase inhibitors identified through structure-based hybridisation.
2003-09-15
Solid-phase synthesis of imidazo[1,2-a]pyridine using sodium benzenesulfinate as a traceless linker.
2002-10-31
Synthesis and biological evaluation of new imidazo[1,2-a]pyridine derivatives designed as mefloquine analogues.
2002-10
Patents
Substance Class Chemical
Created
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Record UNII
G18ZBV2HXA
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Name Type Language
IMIDAZO(1,2-A)PYRIDINE
Preferred Name English
Code System Code Type Description
EPA CompTox
DTXSID80181821
Created by admin on Mon Mar 31 19:51:12 GMT 2025 , Edited by admin on Mon Mar 31 19:51:12 GMT 2025
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FDA UNII
G18ZBV2HXA
Created by admin on Mon Mar 31 19:51:12 GMT 2025 , Edited by admin on Mon Mar 31 19:51:12 GMT 2025
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CAS
274-76-0
Created by admin on Mon Mar 31 19:51:12 GMT 2025 , Edited by admin on Mon Mar 31 19:51:12 GMT 2025
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PUBCHEM
78960
Created by admin on Mon Mar 31 19:51:12 GMT 2025 , Edited by admin on Mon Mar 31 19:51:12 GMT 2025
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