Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Sat Dec 16 12:05:52 GMT 2023
by
admin
on
Sat Dec 16 12:05:52 GMT 2023
|
| Protein Type | ENZYME |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
FMS08T2916
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
Q08499
Created by
admin on Sat Dec 16 12:05:53 GMT 2023 , Edited by admin on Sat Dec 16 12:05:53 GMT 2023
|
PRIMARY | |||
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FMS08T2916
Created by
admin on Sat Dec 16 12:05:53 GMT 2023 , Edited by admin on Sat Dec 16 12:05:53 GMT 2023
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
IC50
|
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INHIBITOR -> TARGET |
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ALLOSTERIC INHIBITOR->TARGET |
Selective negative allosteric modulator with binding affinity values (IC50) of 7.8 nM and 7.4 nM for PDE4D7 and PDE4D3, respectively.
ALLOSTERIC INHIBITOR
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INHIBITOR -> TARGET |
Catalytic domain
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INHIBITOR -> TARGET |
IC50
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RADIOLIGAND->TARGET |
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INHIBITOR->OFF-TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
PDE4D catalytic domain
IC50
|
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
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| Molecular Formula | CHEMICAL |
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