R-138727

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National Institutes of Health Divider Arrow

NCATS

Approval Year

PubMed

PubMed

Title	Date	PubMed
Stereoselective inhibition of human platelet aggregation by R-138727, the active metabolite of CS-747 (prasugrel, LY640315), a novel P2Y12 receptor inhibitor.	2005 Sep	16268477

Substance Class	Mixture Created by `admin` on `Mon Mar 31 22:53:14 GMT 2025` Edited by `admin` on `Mon Mar 31 22:53:14 GMT 2025`
Record UNII	FLN02B3F1J
Record Status	`FAILED`
Record Version

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Name

Type

Language

R-138727 [MI]

Preferred Name

English

R-138727

Common Name

English

(2Z)-2-(1-(2-CYCLOPROPYL-1-(2-FLUOROPHENYL)-2-OXOETHYL)-4-MERCAPTO-3-PIPERIDINYLIDENE) ACETIC ACID

Systematic Name

English

ACETIC ACID, 2-(1-(2-CYCLOPROPYL-1-(2-FLUOROPHENYL)-2-OXOETHYL)-4-MERCAPTO-3-PIPERIDINYLIDENE)-, (2Z)-

Systematic Name

English

Code System Code Type Description

EPA CompTox

DTXSID20699475

Created by admin on Mon Mar 31 22:53:14 GMT 2025 , Edited by admin on Mon Mar 31 22:53:14 GMT 2025

PRIMARY

MERCK INDEX

m9103

Created by admin on Mon Mar 31 22:53:14 GMT 2025 , Edited by admin on Mon Mar 31 22:53:14 GMT 2025

PRIMARY

Merck Index

FDA UNII

FLN02B3F1J

Created by admin on Mon Mar 31 22:53:14 GMT 2025 , Edited by admin on Mon Mar 31 22:53:14 GMT 2025

PRIMARY

CAS

204204-73-9

Created by admin on Mon Mar 31 22:53:14 GMT 2025 , Edited by admin on Mon Mar 31 22:53:14 GMT 2025

PRIMARY

PUBCHEM

10405534

Created by admin on Mon Mar 31 22:53:14 GMT 2025 , Edited by admin on Mon Mar 31 22:53:14 GMT 2025

PRIMARY

All of the following components must be present:


					QP6CO5BO8X

R-125690


					CBH764R26K

R-125687


					N2AQA3AO11

R-125688


					97EDJ67519

R-125689

Related Record Type Details


					G89JQ59I13

PRASUGREL HYDROCHLORIDE

PRODRUG -> METABOLITE ACTIVE


					34K66TBT99

PRASUGREL

PRODRUG -> METABOLITE ACTIVE

Interaction Type:

MAJOR

Qualification:

PLASMA

Amount:

Definition References