AMICARBALIDE DIISETHIONATE

Possibly Marketed Outside US

Details

Stereochemistry	ACHIRAL
Molecular Formula	C15H16N6O.2C2H6O4S
Molecular Weight	548.59
Optical Activity	NONE
Defined Stereocenters	0 / 0
E/Z Centers	0
Charge	0

SHOW SMILES / InChI

Structure Search

SMILES

OCCS(O)(=O)=O.OCCS(O)(=O)=O.NC(=N)C1=CC=CC(NC(=O)NC2=CC=CC(=C2)C(N)=N)=C1

InChI

InChIKey=PWUMRNFCZFZXAE-UHFFFAOYSA-N

InChI=1S/C15H16N6O.2C2H6O4S/c16-13(17)9-3-1-5-11(7-9)20-15(22)21-12-6-2-4-10(8-12)14(18)19;2*3-1-2-7(4,5)6/h1-8H,(H3,16,17)(H3,18,19)(H2,20,21,22);2*3H,1-2H2,(H,4,5,6)

HIDE SMILES / InChI

Molecular Formula	C15H16N6O
Molecular Weight	296.3271
Charge	0
Count

Stereochemistry	ACHIRAL
Additional Stereochemistry	No
Defined Stereocenters	0 / 0
E/Z Centers	0
Optical Activity	NONE

Molecular Formula	C2H6O4S
Molecular Weight	126.132
Charge	0
Count

Stereochemistry	ACHIRAL
Additional Stereochemistry	No
Defined Stereocenters	0 / 0
E/Z Centers	0
Optical Activity	NONE

Description
Sources: https://books.google.ru/books?id=xAPa4WDzAnQC&printsec=frontcover&hl=ru#v=onepage&q&f=false | https://www.ncbi.nlm.nih.gov/pubmed/7216881 | https://www.ncbi.nlm.nih.gov/pubmed/750960

Amicarbalide (Diampron) is an aromatic diamidine exerting piroplasmocidal properties. It is effective against bovine and equine babesiosis and anaplasmosis.

Approval Year

PubMed

Title	Date	PubMed
Cationic antitrypanosomal and other antimicrobial agents in the therapy of experimental Pneumocystis carinii pneumonia.	1988 Jun	3137861
Treatment of experimental pneumocystosis: review of 7 years of experience and development of a new system for classifying antimicrobial drugs.	1992 Sep	1416885
New drug developments for opportunistic infections in immunosuppressed patients: Pneumocystis carinii.	1995 Nov 24	7490723

Substance Class	Chemical Created by `admin` on `Sat Dec 16 08:07:47 GMT 2023` Edited by `admin` on `Sat Dec 16 08:07:47 GMT 2023`
Record UNII	FCC0RF48XI
Record Status	`Validated (UNII)`
Record Version

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Name

Type

Language

AMICARBALIDE DIISETHIONATE

Common Name

English

ETHANESULFONIC ACID, 2-HYDROXY-, COMPD. WITH 3,3'-(CARBONYLDIIMINO)BIS(BENZENECARBOXIMIDAMIDE) (2:1)

Systematic Name

English

AMICARBALIDE DIISETHIONATE [MI]

Common Name

English

M&B-5062A

Code

English

DIAMPRON

Brand Name

English

DIAMPRONE

Brand Name

English

NSC-528032

Code

English

Code System Code Type Description

FDA UNII

FCC0RF48XI