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Details

Stereochemistry ACHIRAL
Molecular Formula C16H15F2N3Si
Molecular Weight 315.3927
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of FLUSILAZOLE

SMILES

C[Si](CN1C=NC=N1)(C2=CC=C(F)C=C2)C3=CC=C(F)C=C3

InChI

InChIKey=FQKUGOMFVDPBIZ-UHFFFAOYSA-N
InChI=1S/C16H15F2N3Si/c1-22(12-21-11-19-10-20-21,15-6-2-13(17)3-7-15)16-8-4-14(18)5-9-16/h2-11H,12H2,1H3

HIDE SMILES / InChI

Molecular Formula C16H15F2N3Si
Molecular Weight 315.3927
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Flusilazole, a member of the demethylation inhibitor fungicides, is highly efficacious for control of fungal infections on a variety of fruit and vegetable crops. Experiments on rodents have shown the marked maternal toxicity, growth retardation, and skeletal abnormalities in the mid- and high-dose groups.

Approval Year

PubMed

PubMed

TitleDatePubMed
Zebrafish embryos as a screen for DNA methylation modifications after compound exposure.
2016-01-15
Combination effects of (tri)azole fungicides on hormone production and xenobiotic metabolism in a human placental cell line.
2014-09-17
Comparison of osteoblast and cardiomyocyte differentiation in the embryonic stem cell test for predicting embryotoxicity in vivo.
2014-09
A high-throughput screen for teratogens using human pluripotent stem cells.
2014-01
Triazole induced concentration-related gene signatures in rat whole embryo culture.
2012-09
Compound-specific effects of diverse neurodevelopmental toxicants on global gene expression in the neural embryonic stem cell test (ESTn).
2012-08-01
Concentration-response analysis of differential gene expression in the zebrafish embryotoxicity test following flusilazole exposure.
2012-05
Chemical class-specific gene expression changes in the zebrafish embryo after exposure to glycol ether alkoxy acids and 1,2,4-triazole antifungals.
2011-09
Discriminating classes of developmental toxicants using gene expression profiling in the embryonic stem cell test.
2011-03-05
Concentration-dependent gene expression responses to flusilazole in embryonic stem cell differentiation cultures.
2011-03-01
Integrated palladium-catalyzed arylation of heavier Group 14 hydrides.
2010-12-03
Determination of fungicides in wine by mixed-mode solid phase extraction and liquid chromatography coupled to tandem mass spectrometry.
2010-11-26
Ecotoxicological effects of rice field waters on selected planktonic species: comparison between conventional and organic farming.
2010-11
Effects of fungicides on in vitro spore germination and mycelial growth of the phytopathogens Leptosphaeria maculans and L. biglobosa (phoma stem canker of oilseed rape).
2010-04
Impact of environmental chemicals on key transcription regulators and correlation to toxicity end points within EPA's ToxCast program.
2010-03-15
Multi-residue analysis of 30 currently used pesticides in fine airborne particulate matter (PM 2.5) by microwave-assisted extraction and liquid chromatography-tandem mass spectrometry.
2009-12-18
In vitro toxicity of selected fungicides from the groups of benzimidazoles and demethylation inhibitors to Cladobotryum dendroides and Agaricus bisporus.
2009-05
Comparison of four different colorimetric and fluorometric cytotoxicity assays in a zebrafish liver cell line.
2008-05-30
Optimization of separation and detection conditions for the multiresidue analysis of pesticides in grapes by comprehensive two-dimensional gas chromatography-time-of-flight mass spectrometry.
2008-05-09
[Occurrence of plant protection product residues in apples in 2007].
2008
Citral, an inhibitor of retinoic acid synthesis, attenuates the frequency and severity of branchial arch abnormalities induced by triazole-derivative fluconazole in rat embryos cultured in vitro.
2007-04-11
Developmental toxic effects of antifungal flusilazole administered by gavage to mice.
2007-02
Comparison of lanosterol-14 alpha-demethylase (CYP51) of human and Candida albicans for inhibition by different antifungal azoles.
2006-11-10
Postulated pathogenic pathway in triazole fungicide induced dysmorphogenic effects.
2006-08
Transferability of six pesticides from agricultural sprayer surfaces.
2006-04
Effects of two systemic fungicides: Artea (Propiconazole+cyproconazole) and Punch (Flusilazole) on the physiology and the respiratory metabolism of durum wheat (Triticum durum L.).
2006
Study on the common teratogenic pathway elicited by the fungicides triazole-derivatives.
2005-09
Pesticide residues on the external surfaces of field crop sprayers: occupational exposure.
2005-06
Determination of azolic fungicides in wine by solid-phase extraction and high-performance liquid chromatography-atmospheric pressure chemical ionization-mass spectrometry.
2005-05-27
Comparative assessment of the inhibition of recombinant human CYP19 (aromatase) by azoles used in agriculture and as drugs for humans.
2004-08
Pesticide residues on the external surfaces of field-crop sprayers: environmental impact.
2004-08
Application of liquid chromatography with electrospray tandem mass spectrometry to the determination of a new generation of pesticides in processed fruits and vegetables.
2004-05-21
Determination of seventeen polar/thermolabile pesticides in apples and apricots by liquid chromatography/mass spectrometry.
2003-07-11
Comparison of microextraction procedures to determine pesticides in oranges by liquid chromatography-mass spectrometry.
2002-09-13
Baseline toxicity of several pesticides to Hyaliodes vitripennis (Say) (Hemiptera: Miridae).
2001-11
Simultaneous determination of six triazolic pesticide residues in apple and pear pulps by liquid chromatography with ultraviolet diode array detection.
2001-10-17
Antifungal triazoles induce malformations in vitro.
2001-08-08
Substance Class Chemical
Created
by admin
on Mon Mar 31 18:54:01 GMT 2025
Edited
by admin
on Mon Mar 31 18:54:01 GMT 2025
Record UNII
F3WG2VVD87
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
NUSTAR
Preferred Name English
FLUSILAZOLE
ISO   MI  
Common Name English
FLUSILAZOLE [MI]
Common Name English
FLUSILAZOLE [ISO]
Common Name English
PUNCH
Brand Name English
BIS(4-FLUOROPHENYL)(METHYL)(1H-1,2,4-TRIAZOL-1-YLMETHYL)SILANE
Systematic Name English
OLYMP
Brand Name English
1-((BIS(4-FLUOROPHENYL)METHYLSILYL)METHYL)-1H-1,2,4-TRIAZOLE
Systematic Name English
FLUZILAZOL
Common Name English
DPX-H6573
Code English
Classification Tree Code System Code
EPA PESTICIDE CODE 128835
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
Code System Code Type Description
PUBCHEM
73675
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY
SMS_ID
300000053334
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY
ALANWOOD
flusilazole
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY
CAS
85509-19-9
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY
CHEBI
81922
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY
WIKIPEDIA
FLUSILAZOLE
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY
MERCK INDEX
m5506
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY Merck Index
FDA UNII
F3WG2VVD87
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY
EPA CompTox
DTXSID3024235
Created by admin on Mon Mar 31 18:54:01 GMT 2025 , Edited by admin on Mon Mar 31 18:54:01 GMT 2025
PRIMARY