Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Sat Dec 16 14:56:33 GMT 2023
by
admin
on
Sat Dec 16 14:56:33 GMT 2023
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
EWR59AZK8G
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
EWR59AZK8G
Created by
admin on Sat Dec 16 14:56:34 GMT 2023 , Edited by admin on Sat Dec 16 14:56:34 GMT 2023
|
PRIMARY | |||
|
Q99250
Created by
admin on Sat Dec 16 14:56:34 GMT 2023 , Edited by admin on Sat Dec 16 14:56:34 GMT 2023
|
PRIMARY | |||
|
Q99250
Created by
admin on Sat Dec 16 14:56:34 GMT 2023 , Edited by admin on Sat Dec 16 14:56:34 GMT 2023
|
PRIMARY |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_212 |
| N | 1_285 |
| N | 1_291 |
| N | 1_297 |
| N | 1_303 |
| N | 1_308 |
| N | 1_340 |
| N | 1_1368 |
| N | 1_1382 |
| N | 1_1393 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
Binds preferentially to Na+ channels in their inactivated state. A high-affinity, stimulus-dependent blocker at the local anesthetic receptor site.
ALLOSTERIC
IC50
|
||
|
INHIBITOR -> TARGET |
EC50
|
||
|
INHIBITOR -> TARGET |
Binds to inactivated state and prevents activation
|
||
|
|
INHIBITOR -> TARGET |
MAY ALSO BLOCK OTHER SODIUM CHANNELS
|
||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|