U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 19:11:33 UTC 2023
Edited
by admin
on Sat Dec 16 19:11:33 UTC 2023
Protein Type RECEPTOR
Protein Sub Type GABA RECEPTOR
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
EV7XZZ7BG9
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
Gamma-aminobutyric acid type B receptor
Common Name English
GABA-B receptor
Common Name English
GABA B receptor
Common Name English
Code System Code Type Description
FDA UNII
EV7XZZ7BG9
Created by admin on Sat Dec 16 19:11:36 UTC 2023 , Edited by admin on Sat Dec 16 19:11:36 UTC 2023
PRIMARY
UNIPROT
O75899
Created by admin on Sat Dec 16 19:11:36 UTC 2023 , Edited by admin on Sat Dec 16 19:11:36 UTC 2023
PRIMARY
UNIPROT
https://www.uniprot.org/uniprot/Q9UBS5
Created by admin on Sat Dec 16 19:11:36 UTC 2023 , Edited by admin on Sat Dec 16 19:11:36 UTC 2023
PRIMARY
From To
1_223 1_260
1_195 1_224
1_66 1_93
2_362 2_396
2_206 2_232
2_117 2_143
2_86 2_131
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_48
N 1_256
N 1_347
N 1_362
N 1_411
N 1_638
N 1_645
N 1_800
N 1_825
N 2_10
N 2_70
N 2_146
N 2_395
N 2_426
N 2_468
N 2_488
N 2_500
N 2_617
Related Record Type Details
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
EC50
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
AGONIST -> TARGET
AGONIST -> TARGET
EC50
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
WEAK AGONIST->TARGET
AGONIST -> TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
Results in enhancement of hippocampal long term potentiation (LTP).
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL