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Details

Stereochemistry MIXED
Molecular Formula C19H30N2O6S
Molecular Weight 414.516
Optical Activity UNSPECIFIED
Defined Stereocenters 0 / 2
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of TISOCROMIDE

SMILES

COC1=CC2=C(C=C1OC)S(=O)(=O)OC(C2)C(=O)NC(C)CC(C)(C)N(C)C

InChI

InChIKey=CXGGLKVQGDLNGH-UHFFFAOYSA-N
InChI=1S/C19H30N2O6S/c1-12(11-19(2,3)21(4)5)20-18(22)16-9-13-8-14(25-6)15(26-7)10-17(13)28(23,24)27-16/h8,10,12,16H,9,11H2,1-7H3,(H,20,22)

HIDE SMILES / InChI

Molecular Formula C19H30N2O6S
Molecular Weight 414.516
Charge 0
Count
Stereochemistry MIXED
Additional Stereochemistry No
Defined Stereocenters 0 / 2
E/Z Centers 0
Optical Activity UNSPECIFIED

Description
Curator's Comment: Description was created based on several sources, including https://www.ncbi.nlm.nih.gov/pubmed/4062921 | https://www.ncbi.nlm.nih.gov/pubmed/262371

Tisocromide exerts antihypoxic and antidepressant action. The details regarding mechanism of action and use are not available.

Approval Year

Conditions

Conditions

ConditionModalityTargetsHighest PhaseProduct
PubMed

PubMed

TitleDatePubMed
Characterization of the antihypoxic activity of tisochromid.
1985
[Antihypoxic effect of tisochromide (16-244) in comparison with piracetam].
1983-04
[Operational evaluation studies in psychopharmacological research (presented with an example of a comparison between clomipramine and tisocromide)].
1980-02
[Comparison of the cardiotoxic effects of tisocromide and imipramine in animal experiment (proceedings)].
1979-05-01
[The clinical effect of a selected sultone (tisocromide) (proceedings)].
1979-05-01
[Tisocromid, a psychopharmaceutical with antidepressive action].
1979
Patents

Sample Use Guides

In Vivo Use Guide
Unknown
Route of Administration: Unknown
In Vitro Use Guide
Unknown
Substance Class Chemical
Created
by admin
on Mon Mar 31 18:06:46 GMT 2025
Edited
by admin
on Mon Mar 31 18:06:46 GMT 2025
Record UNII
ELK0X0H412
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
TISOCROMIDE
INN  
INN  
Official Name English
2,1-BENZOXATHIIN-3-CARBOXAMIDE, N-(3-(DIMETHYLAMINO)-1,3-DIMETHYLBUTYL)-3,4-DIHYDRO-6,7-DIMETHOXY-, 1,1-DIOXIDE
Preferred Name English
N-(3-(DIMETHYLAMINO)-1,3-DIMETHYLBUTYL)-6,7-DIMETHOXY-2,1-BENZOXATHIAN-3-CARBOXAMIDE 1,1-DIOXIDE
Systematic Name English
tisocromide [INN]
Common Name English
Classification Tree Code System Code
NCI_THESAURUS C26170
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
Code System Code Type Description
NCI_THESAURUS
C152662
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
MESH
C022101
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
EPA CompTox
DTXSID10865768
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
ChEMBL
CHEMBL2105495
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
PUBCHEM
65789
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
EVMPD
SUB11120MIG
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
FDA UNII
ELK0X0H412
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
CAS
35423-51-9
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
INN
3241
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
SMS_ID
100000082138
Created by admin on Mon Mar 31 18:06:46 GMT 2025 , Edited by admin on Mon Mar 31 18:06:46 GMT 2025
PRIMARY
Related Record Type Details
ACTIVE MOIETY