Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Wed Apr 02 06:48:22 GMT 2025
by
admin
on
Wed Apr 02 06:48:22 GMT 2025
|
| Protein Type | REGULATOR PROTEIN |
| Protein Sub Type | INITIATION-FACTOR |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
E7D5919XXG
|
| Record Status |
Validated (UNII)
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| Record Version |
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-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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E7D5919XXG
Created by
admin on Wed Apr 02 06:48:22 GMT 2025 , Edited by admin on Wed Apr 02 06:48:22 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
ACTIVATOR -> TARGET |
DNL343 is a selective, orally bioavailable, central nervous system (CNS)–penetrant activator of eukaryotic translation initiation factor 2B (eIF2B).
PRECLINICAL
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO_ACID_SUBSTITUTION | [3_1] | N-TERMINUS | N-ACETYLMETHIONINE | 9J12WX5B6A | ||
| AMINO_ACID_SUBSTITUTION | [1_1] [2_1] | N-TERMINUS | N-ACETYLALANINE | 26C4VY6Z0M | ||
| AMINO_ACID_SUBSTITUTION | [1_18] | SITE_SPECIFIC | TILARGININE | 27JT06E6GR |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
|