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Approval Year

Unknown
139594
Substance Class Protein
Created
by admin
on Sat Dec 16 12:16:39 GMT 2023
Edited
by admin
on Sat Dec 16 12:16:39 GMT 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
DXN1OSB4IB
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
PROGESTERONE RECEPTOR
Common Name English
NUCLEAR RECEPTOR SUBFAMILY 3 GROUP C MEMBER 3
Common Name English
PGR
Common Name English
NR3C3
Common Name English
Code System Code Type Description
UNIPROT
P06401
Created by admin on Sat Dec 16 12:16:41 GMT 2023 , Edited by admin on Sat Dec 16 12:16:41 GMT 2023
PRIMARY
FDA UNII
DXN1OSB4IB
Created by admin on Sat Dec 16 12:16:41 GMT 2023 , Edited by admin on Sat Dec 16 12:16:41 GMT 2023
PRIMARY
Related Record Type Details
Structure of LONAPRISAN
INHIBITOR -> TARGET
Structure of SEGESTERONE
AGONIST -> TARGET
Structure of CHLORMADINONE ACETATE
AGONIST -> TARGET
Twenty times as potent as progesterone as far as its progestational action is concerned
Structure of Progesterone
AGONIST -> TARGET
IC50
Structure of PROMEGESTONE
INHIBITOR -> TARGET
Binding Assay
IC50
Structure of FLUOROFURANYLNORPROGESTERONE F-18
RADIOLIGAND->TARGET
Relative binding affinity (RBA)=190
Structure of TANAPROGET
AGONIST -> TARGET
EC50
Structure of Tanaproget C-11
RADIOLIGAND->TARGET
Structure of TRESTOLONE
AGONIST -> TARGET
Structure of SEGESTERONE ACETATE
AGONIST -> TARGET
EC50
Structure of DIMETHYLTRIENOLONE
AGONIST -> TARGET
Structure of NOMEGESTROL ACETATE
AGONIST -> TARGET
Ki
Structure of DANAZOL
AGONIST -> TARGET
Structure of TELAPRISTONE
INHIBITOR -> TARGET
Structure of ULIPRISTAL
AGONIST -> TARGET
Ulipristal acetate is an orally-active progesterone agonist/antagonist with antagonistic and partial agonistic effects at the progesterone receptor.
BINDING
Structure of BAY-1007626
AGONIST -> TARGET
Structure of VILAPRISAN
MODULATOR->TARGET
Structure of ASOPRISNIL
MODULATOR->TARGET
Structure of DIENOGEST
AGONIST -> TARGET
Structure of CRIDANIMOD
ACTIVATOR OF EXPRESSION->TARGET
Structure of ALLYLESTRENOL
AGONIST -> TARGET
Structure of DIMETHANDROLONE UNDECANOATE
AGONIST -> TARGET
Structure of ULIPRISTAL ACETATE
AGONIST -> TARGET
Structure of CYMIPRISTONE
INHIBITOR -> TARGET
IC50
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
NIH
NCATS
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