U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sun Dec 18 09:30:30 UTC 2022
Edited
by admin
on Sun Dec 18 09:30:30 UTC 2022
Protein Sub Type
Sequence Type COMPLETE
Record UNII
DXN1OSB4IB
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
PROGESTERONE RECEPTOR
Common Name English
NUCLEAR RECEPTOR SUBFAMILY 3 GROUP C MEMBER 3
Common Name English
PGR
Common Name English
NR3C3
Common Name English
Code System Code Type Description
UNIPROT
P06401
Created by admin on Sun Dec 18 09:30:31 UTC 2022 , Edited by admin on Sun Dec 18 09:30:31 UTC 2022
PRIMARY
FDA UNII
DXN1OSB4IB
Created by admin on Sun Dec 18 09:30:31 UTC 2022 , Edited by admin on Sun Dec 18 09:30:31 UTC 2022
PRIMARY
Related Record Type Details
AGONIST -> TARGET
Twenty times as potent as progesterone as far as its progestational action is concerned
RADIOLIGAND->TARGET
Relative binding affinity (RBA)=190
AGONIST -> TARGET
EC50
RADIOLIGAND->TARGET
AGONIST -> TARGET
AGONIST -> TARGET
EC50
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
Ulipristal acetate is an orally-active progesterone agonist/antagonist with antagonistic and partial agonistic effects at the progesterone receptor.
BINDING
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
IC50
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL