U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Thu Jul 06 17:51:08 UTC 2023
Edited
by admin
on Thu Jul 06 17:51:08 UTC 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
DXN1OSB4IB
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
PROGESTERONE RECEPTOR
Common Name English
NUCLEAR RECEPTOR SUBFAMILY 3 GROUP C MEMBER 3
Common Name English
PGR
Common Name English
NR3C3
Common Name English
Code System Code Type Description
UNIPROT
P06401
Created by admin on Thu Jul 06 17:51:10 UTC 2023 , Edited by admin on Thu Jul 06 17:51:10 UTC 2023
PRIMARY
FDA UNII
DXN1OSB4IB
Created by admin on Thu Jul 06 17:51:10 UTC 2023 , Edited by admin on Thu Jul 06 17:51:10 UTC 2023
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
Twenty times as potent as progesterone as far as its progestational action is concerned
AGONIST -> TARGET
IC50
INHIBITOR -> TARGET
Binding Assay
IC50
RADIOLIGAND->TARGET
Relative binding affinity (RBA)=190
AGONIST -> TARGET
EC50
RADIOLIGAND->TARGET
AGONIST -> TARGET
AGONIST -> TARGET
EC50
AGONIST -> TARGET
AGONIST -> TARGET
Ki
AGONIST -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
Ulipristal acetate is an orally-active progesterone agonist/antagonist with antagonistic and partial agonistic effects at the progesterone receptor.
BINDING
AGONIST -> TARGET
MODULATOR->TARGET
MODULATOR->TARGET
AGONIST -> TARGET
ACTIVATOR OF EXPRESSION->TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
IC50
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL