U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 23:28:11 GMT 2025
Edited
by admin
on Tue Apr 01 23:28:11 GMT 2025
Protein Type ENZYME
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
DS8UE5III8
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
GERANYLGERANYL TRANSFERASE
Common Name English
GERANYLGERANYL TRANSFERASE TYPE-1
Preferred Name English
GGTASE-I
Common Name English
GERANYLGERANYLTRANSFERASE TYPE 1
Common Name English
Code System Code Type Description
UNIPROT
P53609
Created by admin on Tue Apr 01 23:28:11 GMT 2025 , Edited by admin on Tue Apr 01 23:28:11 GMT 2025
MAJOR COMPONENT STRUCTURE/SEQUENCE
UNIPROT
P49354
Created by admin on Tue Apr 01 23:28:11 GMT 2025 , Edited by admin on Tue Apr 01 23:28:11 GMT 2025
MAJOR COMPONENT STRUCTURE/SEQUENCE
FDA UNII
DS8UE5III8
Created by admin on Tue Apr 01 23:28:11 GMT 2025 , Edited by admin on Tue Apr 01 23:28:11 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
METAL_BINDING [1_269] [1_271] [1_321] SITE_SPECIFIC ZINC CATION 13S1S8SF37
AMINO_ACID_SUBSTITUTION [2_1] N-TERMINUS N-ACETYLALANINE 26C4VY6Z0M
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL