U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 21:13:26 GMT 2025
Edited
by admin
on Wed Apr 02 21:13:26 GMT 2025
Protein Type MONOCLONAL ANTIBODY
Protein Sub Type IGG4|LAMDA
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
CYQ7L3B6KW
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
Ebrasodebart
INN  
Official Name English
Ent-001
Preferred Name English
ebrasodebart [INN]
Common Name English
immunoglobulin G4-lambda2, anti-[Homo sapiens TMEM219 (transmembrane protein 219, insulin-like growth factor-binding protein 3 receptor, IGFBP-3R) extracellular domain], Homo sapiens monoclonal antibody
Common Name English
Immunoglobulin G4 [226-proline,233-glutamic acid,de-C-terminal-lysine], anti-(human insulin-like growth factor-binding protein 3 receptor) (human monoclonal Ent001 ?4-chain), disulfide with human monoclonal Ent001 ?-chain, dimer
Common Name English
H-gamma4 heavy chain Homo sapiens (1-444) [VH (Homo sapiens IGHV1-18*01 (99.0%) -(IGHD) -IGHJ4*01 (100%), CDR-IMGT [8.8.11](26-33.51-58.97-107)) (1-118)-Homo sapiens IGHG4*01, nG4m(a) CH2 L92, G4v5 h P10, G4v3 CH2 E1.2 (CH1 (119-216), hinge 1-12 S10>P(22
Common Name English
Ent001
Code English
Code System Code Type Description
NCI_THESAURUS
C206903
Created by admin on Wed Apr 02 21:13:26 GMT 2025 , Edited by admin on Wed Apr 02 21:13:26 GMT 2025
PRIMARY
FDA UNII
CYQ7L3B6KW
Created by admin on Wed Apr 02 21:13:26 GMT 2025 , Edited by admin on Wed Apr 02 21:13:26 GMT 2025
PRIMARY
SMS_ID
300000032073
Created by admin on Wed Apr 02 21:13:26 GMT 2025 , Edited by admin on Wed Apr 02 21:13:26 GMT 2025
PRIMARY
INN
12275
Created by admin on Wed Apr 02 21:13:26 GMT 2025 , Edited by admin on Wed Apr 02 21:13:26 GMT 2025
PRIMARY
CAS
2572467-73-1
Created by admin on Wed Apr 02 21:13:26 GMT 2025 , Edited by admin on Wed Apr 02 21:13:26 GMT 2025
PRIMARY
From To
1_22 1_96
2_22 2_96
2_132 4_213
2_145 2_201
2_259 2_319
1_132 3_213
2_365 2_423
3_22 3_87
3_136 3_195
4_22 4_87
4_136 4_195
1_145 1_201
1_224 2_224
1_227 2_227
1_259 1_319
1_365 1_423
Related Record Type Details
ACTIVE MOIETY
anti-(human insulin-like growth factor-binding protein 3 receptor)

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_1] [2_1] [3_1] [4_1] N-TERMINUS Q PIDOLIC ACID SZB83O1W42
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL