U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:44:26 GMT 2025
Edited
by admin
on Tue Apr 01 17:44:26 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
CY360KKS9O
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MYT1
Preferred Name English
MEMBRANE-ASSOCIATED TYROSINE- AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE
Common Name English
MYT1 KINASE
Common Name English
PKMYT1
Common Name English
Code System Code Type Description
WIKIPEDIA
PKMYT1
Created by admin on Tue Apr 01 17:44:26 GMT 2025 , Edited by admin on Tue Apr 01 17:44:26 GMT 2025
PRIMARY
FDA UNII
CY360KKS9O
Created by admin on Tue Apr 01 17:44:26 GMT 2025 , Edited by admin on Tue Apr 01 17:44:26 GMT 2025
PRIMARY
PHAROS
Q99640
Created by admin on Tue Apr 01 17:44:26 GMT 2025 , Edited by admin on Tue Apr 01 17:44:26 GMT 2025
PRIMARY
UNIPROT
Q99640
Created by admin on Tue Apr 01 17:44:26 GMT 2025 , Edited by admin on Tue Apr 01 17:44:26 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
BRET binding assay
IN-VITRO
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_1] M N-ACETYLMETHIONINE 9J12WX5B6A
AMINO ACID SUBSTITUTION [1_40] [1_94] [1_120] [1_143] [1_160] [1_426] [1_469] [1_473] [1_482] S DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_17] [1_495] T THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL