U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 10:25:35 GMT 2025
Edited
by admin
on Wed Apr 02 10:25:35 GMT 2025
Protein Type ENZYME
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
CPW3W3XNP8
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
(PYRUVATE DEHYDROGENASE (ACETYL-TRANSFERRING)) KINASE ISOZYME 1, MITOCHONDRIAL
Common Name English
PDH KINASE 1
Preferred Name English
PDK1 PROTEIN
Common Name English
Pyruvate dehydrogenase kinase 1
Common Name English
PYRUVATE DEHYDROGENASE KINASE ISOFORM 1
Common Name English
PDHK-1
Common Name English
Code System Code Type Description
FDA UNII
CPW3W3XNP8
Created by admin on Wed Apr 02 10:25:35 GMT 2025 , Edited by admin on Wed Apr 02 10:25:35 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_377] SITE_SPECIFIC Amount: N6-SUCCINYLLYSINE 3LH35AJA5L
AMINO_ACID_SUBSTITUTION [1_108] [1_215] [1_216] SITE_SPECIFIC Amount: TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL