U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
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Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:10:37 GMT 2025
Edited
by admin
on Tue Apr 01 18:10:37 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
CE55KZ8SI1
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
TYROSINE-PROTEIN KINASE MER
Common Name English
MER
Preferred Name English
RECEPTOR TYROSINE KINASE MERTK
Common Name English
PROTO-ONCOGENE C-MER
Common Name English
Code System Code Type Description
FDA UNII
CE55KZ8SI1
Created by admin on Tue Apr 01 18:10:37 GMT 2025 , Edited by admin on Tue Apr 01 18:10:37 GMT 2025
PRIMARY
From To
1_95 1_155
1_198 1_242
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_94
N 1_150
N 1_187
N 1_195
N 1_214
N 1_274
N 1_296
N 1_309
N 1_316
N 1_334
N 1_369
N 1_375
N 1_422
N 1_434
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_523] [1_915] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_729] [1_733] [1_734] [1_852] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL