U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 00:55:05 GMT 2025
Edited
by admin
on Wed Apr 02 00:55:05 GMT 2025
Protein Type MONOCLONAL ANTIBODY CONJUGATE
Protein Sub Type IGG1
Sequence Origin HUMANIZED MOUSE
Sequence Type COMPLETE
Record UNII
BPM6YN0KLI
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
BA-3021
Preferred Name English
OZURIFTAMAB VEDOTIN
USAN   INN  
Official Name English
CAB-ROR2-ADC (BA-3021)
Common Name English
BA3021
Code English
Ozuriftamab vedotin [WHO-DD]
Common Name English
OZURIFTAMAB VEDOTIN [USAN]
Common Name English
IMMUNOGLOBULIN G1 (DE-452-LYSINE), ANTI-(HUMAN TYROSINE KINASE RECEPTOR ROR2) (HUMAN-MUS MUSCULUS MONOCLONAL BA302 .GAMMA.1-CHAIN), DISULFIDE WITH HUMAN-MUS MUSCULUS MONOCLONAL BA302 .KAPPA.-CHAIN, DIMER, THIOETHER WITH N-(((4-((N-(6-(3-MERCAPTO-2,5-DIOX
Common Name English
ozuriftamab vedotin [INN]
Common Name English
BA-302 CONJUGATED TO MONOMETHYL AURISTATIN E
Common Name English
Classification Tree Code System Code
FDA ORPHAN DRUG 663018
Created by admin on Wed Apr 02 00:55:05 GMT 2025 , Edited by admin on Wed Apr 02 00:55:05 GMT 2025
Code System Code Type Description
USAN
JK-84
Created by admin on Wed Apr 02 00:55:05 GMT 2025 , Edited by admin on Wed Apr 02 00:55:05 GMT 2025
PRIMARY
NCI_THESAURUS
C155812
Created by admin on Wed Apr 02 00:55:05 GMT 2025 , Edited by admin on Wed Apr 02 00:55:05 GMT 2025
PRIMARY
SMS_ID
300000039974
Created by admin on Wed Apr 02 00:55:05 GMT 2025 , Edited by admin on Wed Apr 02 00:55:05 GMT 2025
PRIMARY
CAS
2460400-11-5
Created by admin on Wed Apr 02 00:55:05 GMT 2025 , Edited by admin on Wed Apr 02 00:55:05 GMT 2025
PRIMARY
INN
11952
Created by admin on Wed Apr 02 00:55:05 GMT 2025 , Edited by admin on Wed Apr 02 00:55:05 GMT 2025
PRIMARY
FDA UNII
BPM6YN0KLI
Created by admin on Wed Apr 02 00:55:05 GMT 2025 , Edited by admin on Wed Apr 02 00:55:05 GMT 2025
PRIMARY
From To
1_22 1_96
2_22 2_96
2_149 2_205
2_225 4_213
2_266 2_326
1_149 1_205
2_372 2_430
3_23 3_87
3_133 3_193
4_23 4_87
4_133 4_193
1_225 3_213
1_231 2_231
1_234 2_234
1_266 1_326
1_372 1_430
Glycosylation Type MAMMALIAN
Glycosylation Link Type Site
N 1_302
N 2_302
Related Record Type Details
ACTIVE MOIETY

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION RESIDUE_SPECIFIC Amount: Cysteinyl vedotin 6603L01WUR
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL