Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Wed Apr 02 07:01:47 GMT 2025
by
admin
on
Wed Apr 02 07:01:47 GMT 2025
|
| Protein Type | RECEPTOR |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
BLL0TO1728
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
BLL0TO1728
Created by
admin on Wed Apr 02 07:01:47 GMT 2025 , Edited by admin on Wed Apr 02 07:01:47 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 3_626 | 3_703 |
| 3_620 | 3_629 |
| 3_613 | 3_616 |
| 3_600 | 3_610 |
| 3_593 | 3_598 |
| 3_572 | 3_579 |
| 3_446 | 3_671 |
| 3_645 | 3_679 |
| 3_561 | 3_570 |
| 3_556 | 3_587 |
| 3_554 | 3_559 |
| 3_535 | 3_540 |
| 3_518 | 3_533 |
| 3_513 | 3_548 |
| 3_511 | 3_516 |
| 3_482 | 3_496 |
| 3_471 | 3_480 |
| 3_466 | 3_505 |
| 3_457 | 3_469 |
| 3_415 | 3_442 |
| 3_28 | 3_55 |
| 3_18 | 3_44 |
| 3_15 | 3_444 |
| 3_7 | 3_25 |
| 2_17 | 2_22 |
| 1_828 | 2_27 |
| 1_677 | 1_690 |
| 1_604 | 1_610 |
| 1_487 | 1_543 |
| 1_151 | 1_164 |
| 1_115 | 1_135 |
| 1_58 | 1_67 |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_43 |
| N | 1_141 |
| N | 1_256 |
| N | 1_266 |
| N | 1_275 |
| N | 1_483 |
| N | 1_489 |
| N | 1_552 |
| N | 1_568 |
| N | 1_634 |
| N | 1_671 |
| N | 1_683 |
| N | 1_732 |
| N | 1_827 |
| N | 3_30 |
| N | 3_74 |
| N | 3_77 |
| N | 3_192 |
| N | 3_249 |
| N | 3_343 |
| N | 3_386 |
| N | 3_397 |
| N | 3_461 |
| N | 3_500 |
| N | 3_649 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
|
INHIBITOR OF ACTIVATION->TARGET |
IC50
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO_ACID_SUBSTITUTION | [3_765] | SITE_SPECIFIC | DEXFOSFOSERINE | VI4F0K069V | ||
| AMINO_ACID_SUBSTITUTION | [3_763] | SITE_SPECIFIC | TYROSINE O-PHOSPHATE | 2R86C98KDX | ||
| AMINO_ACID_SUBSTITUTION | [3_757] [3_769] | SITE_SPECIFIC | THREONINE PHOSPHATE | 3L4WX7B1EI |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
|