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Details

Stereochemistry ABSOLUTE
Molecular Formula C10H13N5O5S
Molecular Weight 315.306
Optical Activity UNSPECIFIED
Defined Stereocenters 4 / 4
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of 8-THIOGUANOSINE

SMILES

NC1=NC2=C(NC(=S)N2[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)C(=O)N1

InChI

InChIKey=KZELNMSPWPFAEB-UMMCILCDSA-N
InChI=1S/C10H13N5O5S/c11-9-13-6-3(7(19)14-9)12-10(21)15(6)8-5(18)4(17)2(1-16)20-8/h2,4-5,8,16-18H,1H2,(H,12,21)(H3,11,13,14,19)/t2-,4-,5-,8-/m1/s1

HIDE SMILES / InChI

Molecular Formula C10H13N5O5S
Molecular Weight 315.306
Charge 0
Count
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 4 / 4
E/Z Centers 0
Optical Activity UNSPECIFIED

Approval Year

PubMed

PubMed

TitleDatePubMed
8-Mercaptoguanosine-mediated enhancement of in vivo IgG1, IgG2 and IgG3 antibody responses to polysaccharide antigens in normal and xid mice.
1989-11-01
8-Mercaptoguanosine overcomes unresponsiveness of human neonatal B cells to polysaccharide antigens.
1988-10-01
Role of salvage and phosphorylation in the immunostimulatory activity of C8-substituted guanine ribonucleosides.
1988-10-01
5-Halo-6-phenyl pyrimidinones and 8-substituted guanosines: biological response modifiers with similar effects on B cells.
1988-03
Activation of human B lymphocytes by 8' substituted guanosine derivatives.
1988-02
Regulation of B-cell differentiation: anti-mu antibodies have opposite effects on differentiation stimulated by bacterial lipopolysaccharide and 8-mercaptoguanosine.
1988
Induction of interleukin 1 activity from macrophages by direct interaction with C8-substituted guanine ribonucleosides.
1988
Inducible Ig heavy chain switching in an IgM+ Ly-1 B cell line. Evidence for a state of switch commitment.
1988
"Numatrin," a nuclear matrix protein associated with induction of proliferation in B lymphocytes.
1987-08-15
Interaction between cytokines and 8-mercaptoguanosine in humoral immunity: synergy with interferon.
1987-07-01
Large, activated B cells are the primary B-cell target of 8-bromoguanosine and 8-mercaptoguanosine.
1987-05
Regulation of B cell activation by prostaglandins: cell cycle-specific effects on activation by anti-immunoglobulin and 8-mercaptoguanosine.
1986-12-15
Distinct effects of dual substitution on inductive and differentiative activities of C8-substituted guanine ribonucleosides.
1986-10-15
Mechanism of synergy between T cell signals and C8-substituted guanine nucleosides in humoral immunity: B lymphotropic cytokines induce responsiveness to 8-mercaptoguanosine.
1986-05-01
Restoration of in vitro responsiveness of xid B cells to TNP-Ficoll by 8-mercaptoguanosine.
1986-02-15
Antigen-specific enhancement of the human antibody response by a substituted nucleoside.
1986
Enhancement of T cell proliferation and differentiation by 8-mercaptoguanosine.
1986
Queuosine metabolism: possible relation to B-cell activation by C8 derivatives of guanosine.
1985-09
Demonstration of T-cell-dependent and T-cell-independent components of 8-mercaptoguanosine-mediated adjuvanticity.
1985-09
Restoration of humoral immunity in vitro in immunodeficient aging mice by C8-derivatized guanine ribonucleosides.
1985-06
Lymphokine-like activity of 8-mercaptoguanosine: induction of T and B cell differentiation.
1985-05
Control of B cell proliferation: inhibition of responses to B cell mitogens induced by plasma cell tumors.
1985-05
Dissociation of inductive from differentiative signals transmitted by C8-substituted guanine ribonucleosides to B cells from SJL mice.
1985-01
Mechanism of 8-mercaptoguanosine-mediated adjuvanticity: roles of clonal expansion and cellular recruitment.
1984-12
Regulation of B-lymphocyte proliferative responses by arachidonate metabolites: effects on membrane-directed versus intracellular activators.
1984-09
Derivatized guanine nucleosides: a new class of adjuvant for in vitro antibody responses.
1983-06
Activation of lymphocytes by a thiol-derivatized nucleoside: characterization of cellular parameters and responsive subpopulations.
1983-02
Patents
Substance Class Chemical
Created
by admin
on Mon Mar 31 19:08:43 GMT 2025
Edited
by admin
on Mon Mar 31 19:08:43 GMT 2025
Record UNII
B0T9FOW56N
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
SQ 12760
Preferred Name English
8-THIOGUANOSINE
Common Name English
GUANOSINE, 7,8-DIHYDRO-8-THIOXO-
Systematic Name English
NSC-79216
Code English
8-MERCAPTOGUANOSINE
Systematic Name English
GUANOSINE, 8-MERCAPTO-
Systematic Name English
Code System Code Type Description
EPA CompTox
DTXSID30948906
Created by admin on Mon Mar 31 19:08:43 GMT 2025 , Edited by admin on Mon Mar 31 19:08:43 GMT 2025
PRIMARY
CAS
686300-03-8
Created by admin on Mon Mar 31 19:08:43 GMT 2025 , Edited by admin on Mon Mar 31 19:08:43 GMT 2025
NON-SPECIFIC STEREOCHEMISTRY
CAS
26001-38-7
Created by admin on Mon Mar 31 19:08:43 GMT 2025 , Edited by admin on Mon Mar 31 19:08:43 GMT 2025
PRIMARY
PUBCHEM
135457302
Created by admin on Mon Mar 31 19:08:43 GMT 2025 , Edited by admin on Mon Mar 31 19:08:43 GMT 2025
PRIMARY
ECHA (EC/EINECS)
247-402-4
Created by admin on Mon Mar 31 19:08:43 GMT 2025 , Edited by admin on Mon Mar 31 19:08:43 GMT 2025
PRIMARY
NSC
79216
Created by admin on Mon Mar 31 19:08:43 GMT 2025 , Edited by admin on Mon Mar 31 19:08:43 GMT 2025
PRIMARY
FDA UNII
B0T9FOW56N
Created by admin on Mon Mar 31 19:08:43 GMT 2025 , Edited by admin on Mon Mar 31 19:08:43 GMT 2025
PRIMARY