U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 01:08:37 GMT 2025
Edited
by admin
on Wed Apr 02 01:08:37 GMT 2025
Protein Type RECEPTOR
Protein Sub Type TYROSINE KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
AA5QJ7X54B
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CD-246 L1196M
Preferred Name English
ANAPLASTIC LYMPHOMA KINASE L1196M
Common Name English
CD246 L1196M
Code English
ALK-L1196M MUTANT
Common Name English
ALK-L1196M CRIZOTINIB RESISTANT MUTANT
Common Name English
ALK L1196M MUTANT
Common Name English
ALK TYROSINE KINASE RECEPTOR L1196M
Systematic Name English
Code System Code Type Description
UNIPROT
Q9UM73
Created by admin on Wed Apr 02 01:08:37 GMT 2025 , Edited by admin on Wed Apr 02 01:08:37 GMT 2025
PRIMARY
FDA UNII
AA5QJ7X54B
Created by admin on Wed Apr 02 01:08:37 GMT 2025 , Edited by admin on Wed Apr 02 01:08:37 GMT 2025
PRIMARY
WIKIPEDIA
ANAPLASTIC LYMPHOMA KINASE
Created by admin on Wed Apr 02 01:08:37 GMT 2025 , Edited by admin on Wed Apr 02 01:08:37 GMT 2025
PRIMARY
EC (ENZYME CLASS)
EC 2.7.10.1
Created by admin on Wed Apr 02 01:08:37 GMT 2025 , Edited by admin on Wed Apr 02 01:08:37 GMT 2025
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_151
N 1_226
N 1_267
N 1_306
N 1_393
N 1_406
N 1_427
N 1_545
N 1_553
N 1_609
N 1_691
N 1_790
N 1_845
N 1_846
N 1_868
N 1_968
Related Record Type Details
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
Ki
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_1060] [1_1074] [1_1078] [1_1113] [1_1260] [1_1489] [1_1586] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL