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Details

Stereochemistry ACHIRAL
Molecular Formula C18H16FN3
Molecular Weight 293.3381
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of FDDNP

SMILES

CN(CCF)C1=CC2=CC=C(C=C2C=C1)C(C)=C(C#N)C#N

InChI

InChIKey=IAVCEBMLYVGBLA-UHFFFAOYSA-N
InChI=1S/C18H16FN3/c1-13(17(11-20)12-21)14-3-4-16-10-18(22(2)8-7-19)6-5-15(16)9-14/h3-6,9-10H,7-8H2,1-2H3

HIDE SMILES / InChI

Molecular Formula C18H16FN3
Molecular Weight 293.3381
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Approval Year

PubMed

PubMed

TitleDatePubMed
Voxel-based analysis of Alzheimer's disease PET imaging using a triplet of radiotracers: PIB, FDDNP, and FDG.
2010-08-15
Dementia mimicking Alzheimer's disease Owing to a tau mutation: CSF and PET findings.
2010-08-05
Quantitative analysis of [18F]FDDNP PET using subcortical white matter as reference region.
2010-03
PET of brain prion protein amyloid in Gerstmann-Sträussler-Scheinker disease.
2010-03
2-(1-{6-[(2-[fluorine-18]fluoroethyl)(methyl) amino]-2-naphthyl} ethylidene)malononitrile (FDDNP) positron emission tomography patterns in nondemented populations.
2010-02
Movement correction method for human brain PET images: application to quantitative analysis of dynamic 18F-FDDNP scans.
2010-02
FDDNP binding using MR derived cortical surface maps.
2010-01-01
Simplified parametric methods for [18F]FDDNP studies.
2010-01-01
Differential association of [11C]PIB and [18F]FDDNP binding with cognitive impairment.
2009-12-15
Relationship of cerebrospinal fluid markers to 11C-PiB and 18F-FDDNP binding.
2009-09
Biomarkers of Alzheimer's disease.
2009-08
Dissecting molecular mechanisms in the living brain of dementia patients.
2009-07-21
Clinical applications of PET amyloid imaging: an update.
2009-07
Depression and anxiety symptoms are associated with cerebral FDDNP-PET binding in middle-aged and older nondemented adults.
2009-06
Differential FDDNP PET patterns in nondemented middle-aged and older adults.
2009-05
Interaction of the amyloid imaging tracer FDDNP with hallmark Alzheimer's disease pathologies.
2009-04
Detection of Alzheimer pathology in vivo using both 11C-PIB and 18F-FDDNP PET.
2009-02
Influence of cognitive status, age, and APOE-4 genetic risk on brain FDDNP positron-emission tomography imaging in persons without dementia.
2009-01
Peripheral metabolism of [(18)F]FDDNP and cerebral uptake of its labelled metabolites.
2008-11
Amyloid imaging in aged and young macaques with [11C]PIB and [18F]FDDNP.
2008-06
[In-vivo imaging of amyloid plaques].
2008-05
Synthesis of 2-(1,1-dicyanopropen-2-yl)-6-(2-[18F]-fluoroethyl)-methylamino-naphthalene ([18F]FDDNP).
2008-02
Limitations of small animal PET imaging with [18F]FDDNP and FDG for quantitative studies in a transgenic mouse model of Alzheimer's disease.
2008-01-18
Evaluation of tracer kinetic models for analysis of [18F]FDDNP studies.
2008-01-14
Amyloid and tau imaging, neuronal losses and function in mild cognitive impairment.
2008-01
Flurbiprofen derivatives in Alzheimer's disease: synthesis, pharmacokinetic and biological assessment of lipoamino acid prodrugs.
2008-01
In vivo molecular imaging biomarkers: clinical pharmacology's new "PET"?
2007-06
PET scanning in mild cognitive impairment.
2007-03-15
PET scanning in mild cognitive impairment.
2007-03-15
Getting a grip on Alzheimer's disease: imaging amyloid in the brain.
2007-03
Seeing what Alzheimer saw.
2007-02
PET of brain amyloid and tau in mild cognitive impairment.
2006-12-21
High-yield, automated radiosynthesis of 2-(1-{6-[(2-[18F]fluoroethyl)(methyl)amino]-2-naphthyl}ethylidene)malononitrile ([18F]FDDNP) ready for animal or human administration.
2006-10-20
The 2,6-disubstituted naphthalene derivative FDDNP labeling reliably predicts Congo red birefringence of protein deposits in brain sections of selected human neurodegenerative diseases.
2006-04
Molecular-imaging probe 2-(1-[6-[(2-fluoroethyl)(methyl) amino]-2-naphthyl]ethylidene) malononitrile labels prion plaques in vitro.
2003-09-03
In vitro detection of (S)-naproxen and ibuprofen binding to plaques in the Alzheimer's brain using the positron emission tomography molecular imaging probe 2-(1-[6-[(2-[(18)F]fluoroethyl)(methyl)amino]-2-naphthyl]ethylidene)malononitrile.
2003
Localization of neurofibrillary tangles and beta-amyloid plaques in the brains of living patients with Alzheimer disease.
2002-01-16
Binding characteristics of radiofluorinated 6-dialkylamino-2-naphthylethylidene derivatives as positron emission tomography imaging probes for beta-amyloid plaques in Alzheimer's disease.
2001-12-15
Patents
Substance Class Chemical
Created
by admin
on Mon Mar 31 22:58:13 GMT 2025
Edited
by admin
on Mon Mar 31 22:58:13 GMT 2025
Record UNII
9U8TYP0V3P
Record Status Validated (UNII)
Record Version
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Name Type Language
PROPANEDINITRILE, 2-(1-(6-((2-FLUOROETHYL)METHYLAMINO)-2-NAPHTHALENYL)ETHYLIDENE)-
Preferred Name English
FDDNP
Common Name English
Code System Code Type Description
FDA UNII
9U8TYP0V3P
Created by admin on Mon Mar 31 22:58:13 GMT 2025 , Edited by admin on Mon Mar 31 22:58:13 GMT 2025
PRIMARY
CAS
590365-47-2
Created by admin on Mon Mar 31 22:58:13 GMT 2025 , Edited by admin on Mon Mar 31 22:58:13 GMT 2025
PRIMARY
PUBCHEM
24858429
Created by admin on Mon Mar 31 22:58:13 GMT 2025 , Edited by admin on Mon Mar 31 22:58:13 GMT 2025
PRIMARY