U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 12:04:38 UTC 2023
Edited
by admin
on Sat Dec 16 12:04:38 UTC 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
9J6QGP7WEA
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ADENOSINE RECEPTOR A1
Common Name English
Adenosine A1
Common Name English
Adenosine A1 receptor
Common Name English
ADORA1
Common Name English
Code System Code Type Description
UNIPROT
P30542
Created by admin on Sat Dec 16 12:04:41 UTC 2023 , Edited by admin on Sat Dec 16 12:04:41 UTC 2023
PRIMARY
FDA UNII
9J6QGP7WEA
Created by admin on Sat Dec 16 12:04:41 UTC 2023 , Edited by admin on Sat Dec 16 12:04:41 UTC 2023
PRIMARY
From To
1_80 1_169
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_159
Related Record Type Details
RADIOLIGAND->TARGET
Ki
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
WEAK INHIBITOR->TARGET
Ki
WEAK INHIBITOR->TARGET
Ki
AGONIST -> TARGET
Ki
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
PARTIAL AGONIST->TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
Binding assay
IC50
INHIBITOR->OFF-TARGET
INHIBITOR -> TARGET
WEAK INHIBITOR->OFF TARGET
Binding Assay
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
PARTIAL AGONIST->TARGET
INHIBITOR -> TARGET
WEAK INHIBITOR->TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR->OFF-TARGET
IC50
LIGAND->TARGET
Kd
INHIBITOR -> TARGET
WEAK INHIBITOR->TARGET
Ki
INHIBITOR -> TARGET
AGONIST -> TARGET
Rat brain receptor
BINDING
Ki
AGONIST -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
Ki
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL