VASOPRESSIN V1A RECEPTOR

Approval Year

Substance Class	Protein
Protein Sub Type
Sequence Type	COMPLETE
Record UNII	9AB783U039
Record Status	`Validated (UNII)`
Record Version

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Name

Type

Language

VASOPRESSIN V1A RECEPTOR

Common Name

English

AVPR1A

Common Name

English

ANTIDIURETIC HORMONE RECEPTOR 1A

Common Name

English

VASCULAR/HEPATIC-TYPE ARGININE VASOPRESSIN RECEPTOR

Common Name

English

AVPR V1A

Common Name

English

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Code System

Code

Type

Description

FDA UNII

9AB783U039

PRIMARY

UNIPROT

P37288

PRIMARY

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Subunit 0

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From	To
1_124	1_203

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Glycosylation Type

HUMAN

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Glycosylation Link Type	Site
N	1_27
N	1_196

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Related Record

Type

Details


					RAX5D5AGV6

BALOVAPTAN

INHIBITOR -> TARGET


					6004MB8Y0D

RIBUVAPTAN

INHIBITOR -> TARGET

Amount:


					GT7UX45K55

Invopressin

PARTIAL AGONIST->TARGET

Comments:

Designed as mixed agonist-antagonist peptide selective for the vasopressin 1a (V1a) receptor with no vasopressin 2 (V2) receptor activity at therapeutic concentrations.

Amount:


					FFM269698K

SKF-100273

INHIBITOR -> TARGET

Interaction Type:

BINDING

Qualification:

IC50

Amount:

0.89 NANOMOLAR (average)


					JJH94R3PWB

NERATINIB

INHIBITOR->OFF-TARGET

Comments:

Radioligand binding assay

Interaction Type:

BINDING

Qualification:

IC50

Amount:

1.1 MICROMOLAR (average)

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Name	Property Type	Amount	Referenced Substance	Defining	Parameters	References
MOL_WEIGHT	CHEMICAL

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