U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 08:17:25 GMT 2025
Edited
by admin
on Wed Apr 02 08:17:25 GMT 2025
Protein Type ENZYME
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
8WC77Y8M4Q
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CYCLIN-DEPENDENT PROTEIN KINASE 5 HOLOENZYME COMPLEX, P35 VARIANT
Common Name English
CDK5/P35 COMPLEX
Preferred Name English
CDK5:P35 COMPLEX
Common Name English
Code System Code Type Description
FDA UNII
8WC77Y8M4Q
Created by admin on Wed Apr 02 08:17:25 GMT 2025 , Edited by admin on Wed Apr 02 08:17:25 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_1] SITE_SPECIFIC N-MYRISTOYLGLYCINE 84UK82T430
AMINO_ACID_SUBSTITUTION [1_137] SITE_SPECIFIC THREONINE PHOSPHATE 3L4WX7B1EI
AMINO_ACID_SUBSTITUTION [1_7] [2_72] [2_159] SITE_SPECIFIC DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL