U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 03:11:43 GMT 2025
Edited
by admin
on Wed Apr 02 03:11:43 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
8UDQ6195SI
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MPS1
Preferred Name English
DUAL SPECIFICITY PROTEIN KINASE TTK
Common Name English
Monopolar Spindle 1
Common Name English
PYT
Common Name English
MPS1L1
Common Name English
PHOSPHOTYROSINE PICKED THREONINE-PROTEIN KINASE
Common Name English
Code System Code Type Description
UNIPROT
P33981
Created by admin on Wed Apr 02 03:11:43 GMT 2025 , Edited by admin on Wed Apr 02 03:11:43 GMT 2025
PRIMARY
FDA UNII
8UDQ6195SI
Created by admin on Wed Apr 02 03:11:43 GMT 2025 , Edited by admin on Wed Apr 02 03:11:43 GMT 2025
PRIMARY
PHAROS
P33981
Created by admin on Wed Apr 02 03:11:43 GMT 2025 , Edited by admin on Wed Apr 02 03:11:43 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Cellular assay
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_33] THREONINE PHOSPHATE 3L4WX7B1EI
AMINO ACID SUBSTITUTION [1_1] N-ACETYLMETHIONINE 9J12WX5B6A
AMINO ACID SUBSTITUTION [1_7] [1_37] [1_80] [1_281] [1_317] [1_321] [1_393] [1_436] [1_821] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL