Details
| Stereochemistry | RACEMIC |
| Molecular Formula | C22H26O3 |
| Molecular Weight | 338.44 |
| Optical Activity | ( + / - ) |
| Defined Stereocenters | 2 / 2 |
| E/Z Centers | 0 |
| Charge | 0 |
SHOW SMILES / InChI
SMILES
CC(C)=C[C@@H]1[C@@H](C(=O)OCC2=COC(CC3=CC=CC=C3)=C2)C1(C)C
InChI
InChIKey=VEMKTZHHVJILDY-UXHICEINSA-N
InChI=1S/C22H26O3/c1-15(2)10-19-20(22(19,3)4)21(23)25-14-17-12-18(24-13-17)11-16-8-6-5-7-9-16/h5-10,12-13,19-20H,11,14H2,1-4H3/t19-,20+/m1/s1
| Molecular Formula | C22H26O3 |
| Molecular Weight | 338.44 |
| Charge | 0 |
| Count |
|
| Stereochemistry | ABSOLUTE |
| Additional Stereochemistry | No |
| Defined Stereocenters | 2 / 2 |
| E/Z Centers | 0 |
| Optical Activity | UNSPECIFIED |
Bioresmethrin is a synthetic pyrethroid insecticide. It is the (+)-trans isomer of resmethrin which itself contains a minimum of 30% bioresmethrin. Bioresmethrin is the [1R, trans] isomer of resmethrin and has greater insecticidal activity than the racemic mixture. Bioresmethrin is a potent contact insecticide effective against a wide range of household insects, plant pests, grain pests and insects found in animal housing. It exhibits a high order of insecticidal activity, which when coupled with its excellent toxicological properties, makes it potentially one of the safest and most useful insecticides now being produced.
CNS Activity
Sources: http://www.t3db.ca/toxins/T3D1844
Curator's Comment: As for every type I pyrethroid, bioresmethrin effects typically include rapid onset of aggressive behavior and increased sensitivity to external stimuli.
Approval Year
PubMed
| Title | Date | PubMed |
|---|---|---|
| Inhibition of carboxylesterase activity of THP1 monocytes/macrophages and recombinant human carboxylesterase 1 by oxysterols and fatty acids. | 2010-01 |
|
| Evidence for dose-additive effects of pyrethroids on motor activity in rats. | 2009-10 |
|
| Pyrethroid insecticides: isoform-dependent hydrolysis, induction of cytochrome P450 3A4 and evidence on the involvement of the pregnane X receptor. | 2009-05-15 |
|
| In vitro metabolism of pyrethroid pesticides by rat and human hepatic microsomes and cytochrome p450 isoforms. | 2009-01 |
|
| Impact of urban agriculture on malaria vectors in Accra, Ghana. | 2008-08-04 |
|
| Susceptibility to thiamethoxam of Musca domestica from Danish livestock farms. | 2008-02 |
|
| Hydrolysis of pyrethroids by human and rat tissues: examination of intestinal, liver and serum carboxylesterases. | 2007-05-15 |
|
| Human carboxylesterases and their role in xenobiotic and endobiotic metabolism. | 2007 |
|
| Identification and quantitation of pyrethroid pesticide residues in vegetables by solid-phase extraction and liquid chromatography/electrospray ionization ion trap mass spectrometry. | 2007 |
|
| Hydrolytic metabolism of pyrethroids by human and other mammalian carboxylesterases. | 2006-02-28 |
|
| Glutathione S-transferase and insecticide resistance in laboratory strains and field populations of Musca domestica. | 2005-08 |
|
| Structure-activity and interaction effects of 14 different pyrethroids on voltage-gated chloride ion channels. | 2004-02 |
|
| Pyrethroid stimulation of ion transport across frog skin. | 2003-06 |
|
| Synergized bifenthrin plus chlorpyrifos-methyl for control of beetles and psocids in sorghum in Australia. | 2003-04 |
|
| Long-term effectiveness of grain protectants and structural treatments against Liposcelis decolor (Pearman) (Psocoptera: Liposcelididae), a pest of stored products. | 2002-12 |
|
| Enzyme-linked immunosorbent assay for the pyrethroid deltamethrin. | 2002-09-25 |
|
| Field studies on the susceptibility of housefly to certain insecticides in nine Egyptian governorates. | 2002-04 |
|
| Enhanced efficiency of electrostatically charged insecticide aerosols. | 2001-05 |
|
| The status and development of insecticide resistance in Danish populations of the housefly Musca domestica L. | 2001-01 |
Patents
Sample Use Guides
2 groups each of 3 rats received i.v. injections into the lateral tail vein of 2.5 mg/kg ([U-14C]phenyl, 2uCi/rat) cismethrin or bioresmethrin as a solution in glycerin formal (3.75 mg/ml).
Route of Administration:
Intravenous
| Substance Class |
Chemical
Created
by
admin
on
Edited
Mon Mar 31 21:00:31 GMT 2025
by
admin
on
Mon Mar 31 21:00:31 GMT 2025
|
| Record UNII |
8535H601Y7
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
DTXSID4091524
Created by
admin on Mon Mar 31 21:00:31 GMT 2025 , Edited by admin on Mon Mar 31 21:00:31 GMT 2025
|
PRIMARY | |||
|
8535H601Y7
Created by
admin on Mon Mar 31 21:00:31 GMT 2025 , Edited by admin on Mon Mar 31 21:00:31 GMT 2025
|
PRIMARY | |||
|
10453-55-1
Created by
admin on Mon Mar 31 21:00:31 GMT 2025 , Edited by admin on Mon Mar 31 21:00:31 GMT 2025
|
PRIMARY |