U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 14:57:49 UTC 2023
Edited
by admin
on Sat Dec 16 14:57:49 UTC 2023
Protein Type RECEPTOR
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
810S9KV11R
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MELANOCORTIN RECEPTOR 1
Common Name English
MC1R
Common Name English
MELANOCYTE-STIMULATING HORMONE RECEPTOR
Common Name English
Code System Code Type Description
UNIPROT
Q01726
Created by admin on Sat Dec 16 14:57:50 UTC 2023 , Edited by admin on Sat Dec 16 14:57:50 UTC 2023
PRIMARY
FDA UNII
810S9KV11R
Created by admin on Sat Dec 16 14:57:50 UTC 2023 , Edited by admin on Sat Dec 16 14:57:50 UTC 2023
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_29
Related Record Type Details
AGONIST -> TARGET
RADIOLIGAND->TARGET
AGONIST -> TARGET
AGONIST -> TARGET
Melanotan II produces melanogenesis by activation of the MC1 receptor.
Ki
WEAK INHIBITOR->TARGET
BINDING
AGONIST -> TARGET
Biased agonist: AP1189 reduced cytokine release but no melanogenesis was induced.
AGONIST -> TARGET
INHIBITOR -> TARGET
Binding assay
Kd
AGONIST -> TARGET
Binding Assay
IC50
AGONIST -> TARGET
Ki
AGONIST -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL