U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 00:41:07 GMT 2025
Edited
by admin
on Wed Apr 02 00:41:07 GMT 2025
Protein Type ENZYME
Protein Sub Type ACYLTRANSFERASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
7U1VP195ST
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
HISTONE ACETYLTRANSFERASE P300
Common Name English
E1A-ASSOCIATED PROTEIN P300
Preferred Name English
HISTONE CROTONYLTRANSFERASE P300
Common Name English
PROTEIN PROPIONYLTRANSFERASE P300
Common Name English
P300 HAT
Common Name English
P300
Common Name English
HISTONE BUTYRYLTRANSFERASE P300
Common Name English
EP300
Common Name English
Code System Code Type Description
NCI_THESAURUS
C17804
Created by admin on Wed Apr 02 00:41:07 GMT 2025 , Edited by admin on Wed Apr 02 00:41:07 GMT 2025
PRIMARY NCIT
FDA UNII
7U1VP195ST
Created by admin on Wed Apr 02 00:41:07 GMT 2025 , Edited by admin on Wed Apr 02 00:41:07 GMT 2025
PRIMARY
EC (ENZYME CLASS)
EC 2.3.1.48
Created by admin on Wed Apr 02 00:41:07 GMT 2025 , Edited by admin on Wed Apr 02 00:41:07 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
METAL_BINDING [1_1743] [1_1747] [1_1752] [1_1757] [1_1766] [1_1770] [1_1778] [1_1781] [1_1791] [1_1795] [1_1800] [1_1805] SITE_SPECIFIC TAZ-TYPE ZINC FINGER FR8G232SRK
AMINO_ACID_SUBSTITUTION [1_1179] [1_1335] [1_1472] [1_1498] [1_1541] [1_1545] [1_1548] [1_1553] [1_1557] [1_1559] [1_1698] [1_1703] [1_1706] SITE_SPECIFIC N6-ACETYLLYSINE 470AD5VY1X
METAL_BINDING [1_1682] [1_1685] [1_1700] [1_1702] SITE_SPECIFIC ZZ-TYPE ZINC FINGER UZ8IXP0HN9
AMINO_ACID_SUBSTITUTION [1_498] SITE_SPECIFIC DEXFOSFOSERINE VI4F0K069V
METAL_BINDING [1_346] [1_350] [1_363] [1_368] [1_377] [1_381] [1_387] [1_392] [1_401] [1_405] [1_410] [1_413] SITE_SPECIFIC TAZ-TYPE ZINC FINGER FR8G232SRK
METAL_BINDING [1_1669] [1_1672] [1_1691] [1_1694] SITE_SPECIFIC ZZ-TYPE ZINC FINGER UZ8IXP0HN9
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL