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Details

Stereochemistry ABSOLUTE
Molecular Formula C24H36O3
Molecular Weight 372.5408
Optical Activity UNSPECIFIED
Defined Stereocenters 6 / 6
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of TESTOSTERONE VALERATE

SMILES

[H][C@@]12CC[C@H](OC(=O)CCCC)[C@@]1(C)CC[C@@]3([H])[C@@]2([H])CCC4=CC(=O)CC[C@]34C

InChI

InChIKey=UCNQPYVHDCHENM-CGRIZKAYSA-N
InChI=1S/C24H36O3/c1-4-5-6-22(26)27-21-10-9-19-18-8-7-16-15-17(25)11-13-23(16,2)20(18)12-14-24(19,21)3/h15,18-21H,4-14H2,1-3H3/t18-,19-,20-,21-,23-,24-/m0/s1

HIDE SMILES / InChI

Molecular Formula C24H36O3
Molecular Weight 372.5408
Charge 0
Count
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 6 / 6
E/Z Centers 0
Optical Activity UNSPECIFIED

Testosterone valerate, or testosterone pentanoate, is a synthetic, steroidal androgen. It is a short-to-medium duration C17β valerate ester of testosterone, with a terminal half-life of approximately twice that of the short-acting testosterone propionate. Testosterone valerate is available exclusively as a component of the veterinary drug Deposterona developed by Syntex Animal Health Company, which is marketed in Mexico. Deposterona also contains testosterone acetate and testosterone undecanoate and is used to treat impotence, weakness, fatigue and hypogonadism in male breeding animals (cows, pigs, canines, sheep), as well as a general protein-sparing anabolic. It is administered via intramuscular injection and acts as a long-lasting prodrug of testosterone. Esterified forms of testosterone are designed to prolong the window of therapeutic effect following administration, allowing for less frequent injection schedule compared to injections of unesterified steroid. Deposterona is also used for bodybuilding purposes in men and not recommended for women performance-enhancing purposes due to its strong androgenic nature, side effects, and slow-acting characteristics (making blood levels difficult to control). Deposterona is only known to be manufactured in Mexico. Because it contains a low concentration of steroid,this product is not in high demand, and not readily diverted for illicit sale.

Approval Year

TargetsConditions

Conditions

ConditionModalityTargetsHighest PhaseProduct
Primary
Deposterona

Approved Use

To treat impotence, weakness, fatigue, and hypogonadism in male breeding animals (cows, pigs, canines, and sheep)
PubMed

PubMed

TitleDatePubMed
Testosterone treatment and 17-ketosteroid excretion. III. Comparison of the time of absorption and excretion of testosterone propionate, testosterone-iso-butyrate, and testosterone-n-valerate.
1952 Jan
Patents

Sample Use Guides

120-360 mg (2-6 ml) Deposterona (12mg of testosterone acetate, 12mg of testosterone valerate, and 36mg of testosterone undecanoate per milliliter of oil) at least weekly for 6-12 weeks for bodybuilding purposes
Route of Administration: Intravascular
In Vitro Use Guide
Unknown
Substance Class Chemical
Created
by admin
on Fri Dec 15 19:42:21 GMT 2023
Edited
by admin
on Fri Dec 15 19:42:21 GMT 2023
Record UNII
7SF23403A0
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
TESTOSTERONE VALERATE
WHO-DD  
Common Name English
Testosterone valerate [WHO-DD]
Common Name English
4-ANDROSTENE-17-.BETA.-OL-3-ONE VALERATE
Common Name English
TESTOSTERONE 17-VALERATE
Common Name English
TESTOSTERONE PENTANOATE
Common Name English
Code System Code Type Description
SMS_ID
100000084797
Created by admin on Fri Dec 15 19:42:21 GMT 2023 , Edited by admin on Fri Dec 15 19:42:21 GMT 2023
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PUBCHEM
102373
Created by admin on Fri Dec 15 19:42:21 GMT 2023 , Edited by admin on Fri Dec 15 19:42:21 GMT 2023
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EVMPD
SUB04746MIG
Created by admin on Fri Dec 15 19:42:21 GMT 2023 , Edited by admin on Fri Dec 15 19:42:21 GMT 2023
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FDA UNII
7SF23403A0
Created by admin on Fri Dec 15 19:42:21 GMT 2023 , Edited by admin on Fri Dec 15 19:42:21 GMT 2023
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CAS
3129-43-9
Created by admin on Fri Dec 15 19:42:21 GMT 2023 , Edited by admin on Fri Dec 15 19:42:21 GMT 2023
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ECHA (EC/EINECS)
221-514-3
Created by admin on Fri Dec 15 19:42:21 GMT 2023 , Edited by admin on Fri Dec 15 19:42:21 GMT 2023
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EPA CompTox
DTXSID40185204
Created by admin on Fri Dec 15 19:42:21 GMT 2023 , Edited by admin on Fri Dec 15 19:42:21 GMT 2023
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WIKIPEDIA
Testosterone valerate
Created by admin on Fri Dec 15 19:42:21 GMT 2023 , Edited by admin on Fri Dec 15 19:42:21 GMT 2023
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