Details
| Stereochemistry | ABSOLUTE |
| Molecular Formula | C16H24N2O3 |
| Molecular Weight | 292.3734 |
| Optical Activity | UNSPECIFIED |
| Defined Stereocenters | 1 / 1 |
| E/Z Centers | 0 |
| Charge | 0 |
SHOW SMILES / InChI
SMILES
CC(C)(C)NC[C@@H](O)COC1=CC=CC2=C1CCC(=O)N2
InChI
InChIKey=LWAFSWPYPHEXKX-LLVKDONJSA-N
InChI=1S/C16H24N2O3/c1-16(2,3)17-9-11(19)10-21-14-6-4-5-13-12(14)7-8-15(20)18-13/h4-6,11,17,19H,7-10H2,1-3H3,(H,18,20)/t11-/m1/s1
| Molecular Formula | C16H24N2O3 |
| Molecular Weight | 292.3734 |
| Charge | 0 |
| Count |
|
| Stereochemistry | ABSOLUTE |
| Additional Stereochemistry | No |
| Defined Stereocenters | 1 / 1 |
| E/Z Centers | 0 |
| Optical Activity | UNSPECIFIED |
(R)-Carteolol is an enantiomer of the drug carteolol that is used to treat glaucoma. (R)-Carteolol is a partial agonist with the high affinity to the beta-adrenoceptors. It was shown, that in the treatment of glaucoma, the therapeutic advantage of the R(+)-isomers is similar to the S(-)-isomers and there is no stereoselectivity between the two enantiomers.
Approval Year
PubMed
| Title | Date | PubMed |
|---|---|---|
| Effects of the R(+)- and S(-)-isomers of beta-adrenoceptor blockers with intrinsic sympathomimetic activity, befunolol and carteolol, on rabbit intraocular pressure. | 1991 Aug |
|
| Comparison of interactions of R-(+)- and S-(-)-isomers of beta-adrenergic partial agonists, befunolol and carteolol, with high affinity site of beta-adrenoceptors in isolated rabbit ciliary body and guinea-pig taenia caeci. | 1991 Jul |
| Substance Class |
Chemical
Created
by
admin
on
Edited
Sat Dec 16 10:56:59 GMT 2023
by
admin
on
Sat Dec 16 10:56:59 GMT 2023
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| Record UNII |
7Q2Q6Q87SS
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| Record Status |
Validated (UNII)
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| Record Version |
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75331-19-0
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7Q2Q6Q87SS
Created by
admin on Sat Dec 16 10:56:59 GMT 2023 , Edited by admin on Sat Dec 16 10:56:59 GMT 2023
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12285397
Created by
admin on Sat Dec 16 10:56:59 GMT 2023 , Edited by admin on Sat Dec 16 10:56:59 GMT 2023
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| Related Record | Type | Details | ||
|---|---|---|---|---|
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RACEMATE -> ENANTIOMER |
