FENPIPALONE

Details

Stereochemistry	RACEMIC
Molecular Formula	C17H22N2O2
Molecular Weight	286.3688
Optical Activity	( + / - )
Defined Stereocenters	0 / 1
E/Z Centers	0
Charge	0

SHOW SMILES / InChI

Structure Search

SMILES

CN1CC(CCN2CCC(=CC2)C3=CC=CC=C3)OC1=O

InChI

InChIKey=YUORBURTMIUPMW-UHFFFAOYSA-N

InChI=1S/C17H22N2O2/c1-18-13-16(21-17(18)20)9-12-19-10-7-15(8-11-19)14-5-3-2-4-6-14/h2-7,16H,8-13H2,1H3

HIDE SMILES / InChI

Molecular Formula	C17H22N2O2
Molecular Weight	286.3688
Charge	0
Count

Stereochemistry	RACEMIC
Additional Stereochemistry	No
Defined Stereocenters	0 / 1
E/Z Centers	0
Optical Activity	( + / - )

Description
Sources: https://www.ncbi.nlm.nih.gov/pubmed/4795993 | https://www.ncbi.nlm.nih.gov/pubmed/4892454

FENPIPALONE is an oxazolidinone derivative with central nervous system depressant and antiinflammatory activity in animal models. However, FENPIPALONE did not demonstrate any usefulness for severely ill chronic schizophrenic patients.

CNS Activity

Approval Year

PubMed

Title	Date	PubMed
Two pilot studies of AHR-1680 in chronic schizophrenic patients.	1969 May-Jun	4892454
5-(2-Aminoethyl)-2-oxazolidinones with central nervous system depressant and antiinflammatory activity.	1973 Oct	4795993

Substance Class	Chemical Created by `admin` on `Sat Dec 16 05:03:40 UTC 2023` Edited by `admin` on `Sat Dec 16 05:03:40 UTC 2023`
Record UNII	6TVC31DEDE
Record Status	`Validated (UNII)`
Record Version

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Name

Type

Language

FENPIPALONE

Official Name

English

3-METHYL-5-(2-(4-PHENYL-1,2,3,6-TETRAHYDRO-1-PYRIDYL)ETHYL)-2-OXAZOLIDINONE

Systematic Name

English

fenpipalone [INN]

Common Name

English

FENPIPALONE [USAN]

Common Name

English

AHR-1680

Code

English

5-[2-(3,6-Dihydro-4-phenyl-1(2H)-pyridyl)ethyl]-3-methyl-2-oxazolidinone

Systematic Name

English

2-OXAZOLIDINONE, 5-(2-(3,6-DIHYDRO-4-PHENYL-1(2H)-PYRIDINYL)ETHYL)-3-METHYL-

Systematic Name

English

Classification Tree Code System Code

NCI_THESAURUS

C257