U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
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Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:50:57 GMT 2025
Edited
by admin
on Tue Apr 01 16:50:57 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
6OU487748Q
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
SUBSTANCE-P RECEPTOR
Common Name English
NEUROKININ-1 RECEPTOR
Preferred Name English
TACHYKININ RECEPTOR 1
Common Name English
NK-1 RECEPTOR
Common Name English
TACR1
Common Name English
NK1 RECEPTOR
Common Name English
NK1R
Common Name English
Code System Code Type Description
FDA UNII
6OU487748Q
Created by admin on Tue Apr 01 16:50:57 GMT 2025 , Edited by admin on Tue Apr 01 16:50:57 GMT 2025
PRIMARY
WIKIPEDIA
Tachykinin receptor 1
Created by admin on Tue Apr 01 16:50:57 GMT 2025 , Edited by admin on Tue Apr 01 16:50:57 GMT 2025
PRIMARY
PHAROS
P25103
Created by admin on Tue Apr 01 16:50:57 GMT 2025 , Edited by admin on Tue Apr 01 16:50:57 GMT 2025
PRIMARY
UNIPROT
P25103
Created by admin on Tue Apr 01 16:50:57 GMT 2025 , Edited by admin on Tue Apr 01 16:50:57 GMT 2025
PRIMARY
From To
1_105 1_180
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_14
N 1_18
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> 200-fold selectivity against NK2 and NK3 receptors
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INHIBITOR->OFF-TARGET
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Percent inhibition of specific binding
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HUMAN IM CELLS
BINDING
Ki
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NON-INHIBITOR->OFF TARGET
IC50
RADIOLIGAND->TARGET
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INHIBITOR -> TARGET
INHIBITOR -> TARGET
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ANTAGONIST
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Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL