U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:46:41 GMT 2025
Edited
by admin
on Tue Apr 01 18:46:41 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
6N29KC6F1M
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 2
Common Name English
ERK ACTIVATOR KINASE 2
Preferred Name English
MAPK/ERK KINASE 2
Common Name English
MAPKK 2
Common Name English
MAP KINASE KINASE 2
Common Name English
MAP2K2
Common Name English
Code System Code Type Description
FDA UNII
6N29KC6F1M
Created by admin on Tue Apr 01 18:46:41 GMT 2025 , Edited by admin on Tue Apr 01 18:46:41 GMT 2025
PRIMARY
PHAROS
P36507
Created by admin on Tue Apr 01 18:46:41 GMT 2025 , Edited by admin on Tue Apr 01 18:46:41 GMT 2025
PRIMARY
UNIPROT
P36507
Created by admin on Tue Apr 01 18:46:41 GMT 2025 , Edited by admin on Tue Apr 01 18:46:41 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
UNCOMPETITIVE
INHIBITOR -> TARGET
IN-VITRO
INHIBITOR -> TARGET
competitive with ATP increases in ATP led to increased IC50. Value for 1 micromolar ATP
REVERSIBLE
IC50
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_222] [1_226] S O-ACETYLSERINE G05L7T7ZEQ
AMINO ACID SUBSTITUTION [1_222] S DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL