Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 18:46:41 GMT 2025
by
admin
on
Tue Apr 01 18:46:41 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
6N29KC6F1M
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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6N29KC6F1M
Created by
admin on Tue Apr 01 18:46:41 GMT 2025 , Edited by admin on Tue Apr 01 18:46:41 GMT 2025
|
PRIMARY | |||
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P36507
Created by
admin on Tue Apr 01 18:46:41 GMT 2025 , Edited by admin on Tue Apr 01 18:46:41 GMT 2025
|
PRIMARY | |||
|
P36507
Created by
admin on Tue Apr 01 18:46:41 GMT 2025 , Edited by admin on Tue Apr 01 18:46:41 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
UNCOMPETITIVE
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|
INHIBITOR -> TARGET |
IN-VITRO
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INHIBITOR -> TARGET |
competitive with ATP increases in ATP led to increased IC50. Value for 1 micromolar ATP
REVERSIBLE
IC50
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INHIBITOR -> TARGET |
IC50
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_222] [1_226] | S | O-ACETYLSERINE | G05L7T7ZEQ | ||
| AMINO ACID SUBSTITUTION | [1_222] | S | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|