U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 12:54:26 UTC 2023
Edited
by admin
on Sat Dec 16 12:54:26 UTC 2023
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
6KTD5QW2LA
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
GAMMA-AMINOBUTYRIC ACID TYPE B RECEPTOR SUBUNIT 1
Common Name English
GABA-BR1
Common Name English
GABABR1
Common Name English
GABA-B RECEPTOR 1
Common Name English
GPRC3A
Common Name English
Code System Code Type Description
FDA UNII
6KTD5QW2LA
Created by admin on Sat Dec 16 12:54:26 UTC 2023 , Edited by admin on Sat Dec 16 12:54:26 UTC 2023
PRIMARY
UNIPROT
Q9UBS5
Created by admin on Sat Dec 16 12:54:26 UTC 2023 , Edited by admin on Sat Dec 16 12:54:26 UTC 2023
PRIMARY
From To
1_86 1_131
1_117 1_143
1_206 1_232
1_362 1_396
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_10
N 1_70
N 1_395
N 1_426
N 1_468
N 1_488
N 1_500
Related Record Type Details
AGONIST -> TARGET
Binding assay
IC50
AGONIST -> TARGET
Binding Assay
IC50
INHIBITOR -> TARGET
Binding Assay
IC50
AGONIST -> TARGET
It is less potent as a GABAB receptor agonist than baclofen but more potent than phenibut.
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL