U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
This repository is under review for potential modification in compliance with Administration directives.

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:06:15 GMT 2025
Edited
by admin
on Tue Apr 01 17:06:15 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
6EM0N6I9ZP
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
PROSTANOID EP4 RECEPTOR
Preferred Name English
PROSTAGLANDIN E2 RECEPTOR EP4 SUBTYPE
Common Name English
PTGER4
Common Name English
Code System Code Type Description
FDA UNII
6EM0N6I9ZP
Created by admin on Tue Apr 01 17:06:15 GMT 2025 , Edited by admin on Tue Apr 01 17:06:15 GMT 2025
PRIMARY
UNIPROT
P35408
Created by admin on Tue Apr 01 17:06:15 GMT 2025 , Edited by admin on Tue Apr 01 17:06:15 GMT 2025
PRIMARY
From To
1_92 1_170
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_7
Related Record Type Details
WEAK AGONIST->TARGET
Ki
AGONIST -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
RADIOLIGAND->TARGET
Kd
AGONIST -> TARGET
IC50
WEAK AGONIST->TARGET
Ki
AGONIST -> TARGET
AGONIST -> TARGET
Ki
INHIBITOR -> TARGET
Ki
INHIBITOR -> TARGET
AGONIST -> TARGET
Ki
INHIBITOR -> TARGET
Human EP4 receptor-expressing Jurkat cells.
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_374] [1_377] [1_379] [1_382] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL