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Details

Stereochemistry ACHIRAL
Molecular Formula C24H23F2NO4
Molecular Weight 427.4405
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of FEDAA-1106

SMILES

COC1=CC(CN(C(C)=O)C2=C(OC3=CC=CC=C3)C=CC(F)=C2)=C(OCCF)C=C1

InChI

InChIKey=NZVKWLWAFUSDQE-UHFFFAOYSA-N
InChI=1S/C24H23F2NO4/c1-17(28)27(16-18-14-21(29-2)9-11-23(18)30-13-12-25)22-15-19(26)8-10-24(22)31-20-6-4-3-5-7-20/h3-11,14-15H,12-13,16H2,1-2H3

HIDE SMILES / InChI

Molecular Formula C24H23F2NO4
Molecular Weight 427.4405
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

FEDAA1106 (N-(5-fluoro-2-phenoxyphenyl)-N-(2-(2-fluoroethoxy)-5-methoxybenzyl) acetamide) is a selective ligand for TSPO-18kDa (also known as peripheral benzodiazepine receptor). Radiolabeled 18F FEDAA1106 is a PET tracer. Imaging the 18-kDa translocator protein (TSPO) is considered a potential tool for in vivo evaluation of macrophage activation and inflammation.

Approval Year

Substance Class Chemical
Created
by admin
on Mon Mar 31 22:10:01 GMT 2025
Edited
by admin
on Mon Mar 31 22:10:01 GMT 2025
Record UNII
684F91Q1TR
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
FEDAA-1106
Common Name English
FEDAA1106
Preferred Name English
ACETAMIDE, N-((2-(2-FLUOROETHOXY)-5-METHOXYPHENYL)METHYL)-N-(5-FLUORO-2-PHENOXYPHENYL)-
Systematic Name English
Code System Code Type Description
FDA UNII
684F91Q1TR
Created by admin on Mon Mar 31 22:10:01 GMT 2025 , Edited by admin on Mon Mar 31 22:10:01 GMT 2025
PRIMARY
CAS
505084-41-3
Created by admin on Mon Mar 31 22:10:01 GMT 2025 , Edited by admin on Mon Mar 31 22:10:01 GMT 2025
PRIMARY
PUBCHEM
9845414
Created by admin on Mon Mar 31 22:10:01 GMT 2025 , Edited by admin on Mon Mar 31 22:10:01 GMT 2025
PRIMARY